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N-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-(prop-2-yn-1-yl)cyclohexanamine
1-(3-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}phenyl)ethan-1-one
1-[(2-chlorophenyl)methyl]-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
1-(1-benzothiophen-5-ylmethyl)-4-[2-(methylsulfanyl)propyl]-1H-1,2,3-triazole
2-(2-methoxyethyl)-8-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
2-(phenoxathiin-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N,5-dimethyl-1-propyl-N-(quinolin-5-ylmethyl)-1H-pyrazole-4-carboxamide
N-(4-chloro-2-ethylphenyl)-3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazine-1-carboxamide
3-[6-(azepan-1-yl)pyridazin-3-yl]benzoic acid
7-[3-(4-methylphenyl)propanoyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N3-cyclohexyl-N5-[2-(1H-indol-3-yl)ethyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]-N-(1,3-thiazol-2-yl)propanamide
N-methyl-N-(1-{1-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
N-(2-fluorophenyl)-5-(1H-pyrazol-4-yl)furan-2-carboxamide
(2S)-3-(4-hydroxyphenyl)-2-[(2-methyl-1-benzofuran-7-yl)formamido]propanamide
3-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-1-(propan-2-yl)piperidine
3-(2,3-dihydro-1-benzofuran-7-yl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
4-{3-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]phenyl}-4H-1,2,4-triazole
2-amino-4-(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
3-(4-methoxyphenyl)-N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-1H-pyrazole-5-carboxamide
N-({2-[(4-methoxyphenyl)methyl]-6-oxo-1,6-dihydropyrimidin-4-yl}methyl)furan-3-carboxamide
N-methyl-N-[(1S)-1-phenylethyl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
3-(pyridin-2-ylmethoxy)-N-[3-(4H-1,2,4-triazol-4-yl)phenyl]piperidine-1-carboxamide
3-[(4-acetamidophenyl)methyl]-N-[(3-fluorophenyl)methyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-(2-{1-[(3,5-dichloropyridin-4-yl)methyl]piperidin-2-yl}ethyl)morpholine
{[3-(4-fluorophenyl)oxolan-3-yl]methyl}(methyl)(thiophen-2-ylmethyl)amine
5-{[(2,6-difluoro-3-methylphenyl)methyl]amino}-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-[4-(dimethylamino)azepan-1-yl]ethan-1-one
1-[3-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)benzenesulfonyl]-1,4-diazepane
1-{[2-(difluoromethoxy)phenyl]methyl}-N-(3,4-dimethoxyphenyl)piperidin-3-amine
4-{[4-(adamantan-1-yl)piperazin-1-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile
2-butyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-1,3-benzoxazole-5-carboxamide
3-{[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]methyl}benzonitrile
2-[3-(1H-pyrazol-3-yl)phenyl]-6-(pyrrolidine-1-carbonyl)pyrazine
1-[(1-benzyl-1H-indol-6-yl)methyl]-4-(hydroxymethyl)azepan-4-ol
2-{4-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}-1,3-benzothiazole
3,3,3-trifluoro-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
1-(2-methyl-1,3-thiazole-4-carbonyl)-3-[(methylsulfanyl)methyl]piperidine
[(3R,4R)-4-[(dimethylamino)methyl]-1-(5-methylthiophene-3-carbonyl)pyrrolidin-3-yl]methanol
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-ethyl-4-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
1-methyl-4-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-[(2,3-dimethoxyphenyl)methyl]-N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[2-(dimethylamino)ethyl]-N-[(3-methylthiophen-2-yl)methyl]-1H-indole-2-carboxamide
1-(3-ethyl-1,2-oxazole-5-carbonyl)-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]benzene-1-sulfonamide
1-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-{[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}azocane
(3R,4R)-3-methyl-1-(1-methyl-1H-pyrazole-4-carbonyl)-4-(oxan-4-yl)piperidin-4-ol
5-methanesulfonyl-1'-(3-methyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]