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N-{[1-(4-methanesulfonylbenzenesulfonyl)piperidin-3-yl]methyl}thiophene-2-carboxamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}[(4-methoxyphenyl)methyl](oxolan-2-ylmethyl)amine
3-cyclopropyl-N-methyl-N-[(3-methylthiophen-2-yl)methyl]-1H-pyrazole-5-carboxamide
5-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-N,4-dimethyl-1,3-thiazol-2-amine
(1S,4S)-2-{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}-2-azabicyclo[2.2.1]heptane
N-ethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
8-(2,3-dihydro-1H-inden-2-yl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-{4-[(butylsulfanyl)methyl]-5-methylfuran-2-carbonyl}-2-(trifluoromethyl)morpholine
9-(2-methyl-1H-pyrrole-3-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(4-methyl-1,3-thiazol-5-yl)-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)propanamide
2-(4-carbamoylpiperidin-1-yl)-2-[2-(methylsulfanyl)phenyl]acetic acid
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
4-(naphthalen-2-ylmethyl)-3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]piperazin-2-one
3-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]benzonitrile
3-hydroxy-3-({[2-(1-hydroxycyclopentyl)ethyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
ethyl 2-[2-(pyridin-2-yl)pyrrolidin-1-yl]acetate
2,2-bis(hydroxymethyl)-1-{2-methyl-2,7-diazaspiro[4.5]decan-7-yl}butan-1-one
(3aS,6aR)-3-[3-(4-methoxyphenyl)propyl]-2-oxo-N-(propan-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-1-ethyl-3-methylpiperidine-3-carboxamide
2,6-di-tert-butyl-4-[3-(hydroxymethyl)-4-methylpiperazine-1-carbonyl]phenol
2-(2H-1,3-benzodioxol-5-yloxy)-1-[3-methyl-4-(propan-2-yl)piperazin-1-yl]ethan-1-one
N-methyl-2-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-4-yl}acetamide
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidine-4-carboxylic acid
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(2-hydroxyacetyl)pyrrolidine-3-carboxylic acid
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(ethyl)(2-methoxyethyl)amine
1-(azepan-1-yl)-3-[3-({[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]propan-2-ol
(1S,5R)-3-benzoyl-6-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(2-{1-oxa-8-azaspiro[4.6]undecan-8-yl}-2-oxoethyl)-1,2-dihydroquinoxalin-2-one
ethyl 4-(1-{4-[(1-phenylethyl)carbamoyl]phenyl}piperidin-4-yl)piperazine-1-carboxylate
3-hexyl-8-(5-hydroxypyrazine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})(pyridin-4-ylmethyl)amine
4-[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-methyl-2-oxo-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,2-dihydroquinoline-3-carboxamide
(3R,4R)-1-[(6-chloro-2H-chromen-3-yl)methyl]-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-1-(4-methylpiperidin-1-yl)propan-1-one
2-{3-[2-(3-methoxyphenyl)ethyl]piperidine-1-carbonyl}pyridine
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-(2-methylpropyl)-1,3-oxazole-4-carboxamide
[(3R,4S)-1-[(3-chloro-4-fluorophenyl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
(1S,5R)-3-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(2,6-dimethylpyridin-3-yl)-N-[(1-ethylpiperidin-2-yl)methyl]pyrimidin-2-amine
2-{[(3,5-dimethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]amino}-N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)acetamide
3-(azepane-1-carbonyl)-1-ethyl-N-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(cyclopropylmethyl)-4-[2-(1H-pyrazol-1-yl)benzoyl]piperazine
N-[(3-chloro-1-benzothiophen-2-yl)methyl]-4-hydroxy-N,2-dimethylpyrimidine-5-carboxamide
(2S,4S,5R)-5-(2-chlorophenyl)-1,2-dimethyl-4-(4-methylpiperazine-1-carbonyl)pyrrolidine-2-carboxylic acid
3-phenyl-8-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-1,8-diazaspiro[4.5]decan-2-one
N-[(2-chlorophenyl)methyl]-N-cyclopropyl-3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanamide
1-({5-[1-(3-fluoropyridin-4-yl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
2-{4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol