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1-cyclohexyl-3-(cyclopropylmethyl)-N-(1H-imidazol-2-ylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-(4-chlorophenoxy)-1-[(3S,7S)-3-(hydroxymethyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-5-yl]ethan-1-one
1-cyclopentanecarbonyl-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]piperidine-4-carboxamide
5-methyl-3-[3-(4-methyl-3-oxopiperazin-1-yl)-3-oxopropyl]-2,3-dihydro-1,3-benzoxazol-2-one
1-ethyl-5-{4-phenyl-1-[2-(thiophen-2-yl)ethyl]-1H-imidazol-5-yl}-1H-1,2,4-triazole
methyl 2-({4-[1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-5-(4-fluorophenyl)pyrimidin-2-yl}sulfanyl)acetate
1-[2-(2,2-diphenylethyl)morpholin-4-yl]-2-(furan-2-yl)ethane-1,2-dione
5-[1-methyl-5-(morpholin-4-yl)-1H-1,2,4-triazol-3-yl]pyridin-3-amine
1-(pyrrolidine-1-sulfonyl)-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazine
3-(1H-1,3-benzodiazol-1-yl)-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]propan-1-one
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]pent-4-en-1-one
5-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]pentanamide
5-[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]-1-propyl-1H-pyrazole
1-[(3,4-dimethoxyphenyl)methyl]-3-[3-(propan-2-yloxy)benzoyl]piperidine
1-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-{2-[(3,5-dimethyladamantan-1-yl)oxy]ethyl}-2-(1H-imidazol-4-yl)-1H-imidazole
N-benzyl-N-ethyl-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
3-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-4-yl}-1-(piperidin-4-ylmethyl)urea
3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-(pyridin-3-ylmethyl)propanamide
8-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-6-(propan-2-yl)pyridine-3-carbonitrile
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}butanamide
N-{[3-methyl-7-(4-phenylbenzoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1,3-thiazole-5-carboxamide
3-(4-methoxy-3,5-dimethylbenzoyl)-1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidine
1-(6-cyclopropylpyrimidin-4-yl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-[2-(methylamino)pyridine-4-carbonyl]-1,4-diazepan-6-ol
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-1-(3-propanoylpiperidin-1-yl)propan-1-one
6-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-2-carbonitrile
8-(1,3-benzoxazol-2-yl)-1-[(2-ethylpyrimidin-5-yl)methyl]-1,8-diazaspiro[4.5]decane
{[2-(3-chlorophenyl)-6,7-dimethoxyquinolin-3-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}acetamide
ethyl 1-[(5-ethylthiophen-2-yl)sulfonyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
2-methyl-6-[2-(pyridin-4-yl)quinoline-4-carbonyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-methyl-N-(oxan-4-yl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
2-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(pyridin-4-ylmethyl)amino)butan-1-ol
N-(1-ethyl-1H-1,2,4-triazol-3-yl)-3-(2-hydroxypropan-2-yl)piperidine-1-carboxamide
6-methyl-3-[2-(trifluoromethyl)morpholine-4-carbonyl]-1,4-dihydroquinolin-4-one
(2S)-2-(methoxymethyl)-N-[2-(piperidin-1-ylmethyl)phenyl]pyrrolidine-1-carboxamide
1-[(3-chlorophenyl)methyl]-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperazine
2-(2-aminoethyl)-N-[2-(4-methylpiperazin-1-yl)butyl]quinazolin-4-amine
N-({8-benzyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-(morpholin-4-yl)propanamide
N-[(4-methoxy-2,5-dimethylphenyl)methyl]-N-methyloxan-4-amine
1-(3-chlorophenyl)-5-methyl-4-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperazin-2-one
[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl](benzyl)[(4-methyl-1,3-thiazol-5-yl)methyl]amine
(4aR,8aR)-2-cyclopentanecarbonyl-7-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-decahydro-2,7-naphthyridin-4a-ol
(1-methoxypropan-2-yl)({[4-(1H-pyrazol-3-yl)phenyl]methyl})amine
4-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}benzenesulfonyl)morpholine
N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)-1,3-thiazole-5-carboxamide
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-{[1-(propan-2-yl)piperidin-4-yl]methyl}propanamide
1-[4-(4-aminopyrimidin-2-yl)-6-hydroxy-1,4-diazepan-1-yl]ethan-1-one