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(1S,5R)-3-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(3-hydroxy-3-phenylpropyl)-N-methyl-2-(methylamino)pyridine-4-carboxamide
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(2-methoxyethyl)-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
5-(4-{1-[N-methyl-1-(2-methylfuran-3-yl)formamido]-2-phenylethyl}piperidine-1-carbonyl)-2,1,3-benzoxadiazol-1-ium-1-olate
1-(4-{5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-diazepan-1-yl)ethan-1-one
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-[(6-methylpyridin-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{[2-methoxy-5-(pyridin-4-yl)phenyl]methyl}cyclopentanamine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
(1R,2S)-N1-butyl-N2-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]cyclohexane-1,2-dicarboxamide
8-(butan-2-yl)-1-methyl-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 4-(cyclopropylmethyl)-1-[2-(2H-indazol-2-yl)acetyl]piperidine-4-carboxylate
N-{[5-fluoro-7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-methyl-1,3-oxazole-5-carboxamide
5-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}-N-(propan-2-yl)pyrimidin-2-amine
3-[(3R,4S)-4-(morpholin-4-yl)-1-(5-phenyl-1,3,4-thiadiazol-2-yl)piperidin-3-yl]propanoic acid
2-(3-cyclopentyl-5-{5-methylimidazo[1,2-a]pyridin-2-yl}-1H-1,2,4-triazol-1-yl)ethan-1-ol
5-[1-(benzenesulfonyl)cyclopropyl]-3-cyclopropyl-1-phenyl-1H-1,2,4-triazole
N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-4-(4H-1,2,4-triazol-4-yl)benzamide
(3aR,6aR)-2-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-{2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-oxo-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-[(2-phenoxypyridin-3-yl)methyl]but-3-enamide
4-[1-({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)piperidin-4-yl]pyridine
5-cyclopropyl-3-{[5-(2-methyl-1,3-thiazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
3-methyl-N-[(5-methylpyrazin-2-yl)methyl]-4-oxo-3,4-dihydroquinazoline-7-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
3-(4-{2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]ethyl}-1,3-thiazol-2-yl)pyridine
(2S,4S)-4-amino-1-(3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}propanoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
3,3-dimethyl-1-[(3S,4R)-1-{2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl}-4-(propan-2-yl)pyrrolidin-3-yl]urea
1-cyclopropyl-4-{[2-(2-methyl-1-benzothiophen-3-yl)-1H-imidazol-1-yl]methyl}pyrrolidin-2-one
4-[2-(4-fluorophenyl)azetidine-1-carbonyl]-2-propyl-1,3-thiazole
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-methylacetamide
N-[(3S,4R)-1-[2-(2H-indazol-2-yl)acetyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
2-(1H-indazol-1-yl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}acetamide
6-{4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-9H-purine
3-chloro-N-cyclopentyl-4-({1-[3-(methylsulfanyl)propyl]piperidin-4-yl}oxy)benzamide
1-cycloheptyl-N-[(6-methylpyridin-2-yl)methyl]-6-oxopiperidine-3-carboxamide
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-(2,2-dimethylpropyl)piperidine
(1S,5R)-6-(2-methoxyethyl)-3-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(3R,4R)-1-(3-chloro-4-methoxybenzenesulfonyl)-3,4-dimethylpyrrolidin-3-ol
methyl 3-[4-(4-hydroxypiperidin-1-yl)piperidine-1-carbonyl]-5-methoxybenzoate
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}ethan-1-one
(4aS,8aR)-1-propyl-6-[3-(pyridin-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
2-cyclopropyl-5-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-4-methylpyrimidine
1-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-ethylpiperidin-3-ol
N-{[4-(piperidine-1-carbonyl)phenyl]methyl}-4-(pyridin-3-yl)pyrimidin-2-amine
2-amino-6-cyclopropyl-4-{2-[2-(morpholin-4-yl)ethoxy]phenyl}pyridine-3-carbonitrile
1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(1H-1,2,3-triazole-5-carbonyl)-1,4-diazepan-6-ol
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-5-[4-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}cyclopropan-1-amine
(3R,4R)-4-(azepan-1-yl)-1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-3-ol