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3-(4-methoxyphenyl)-3-phenyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}propanamide
3-[(3R,4S)-4-(dimethylamino)-1-(1-methyl-5-phenyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]propanoic acid
1-[2-(3-fluorophenyl)ethyl]-N-methyl-N-[(3-methylpyridin-2-yl)methyl]-6-oxopiperidine-3-carboxamide
3-{1-[4-hydroxy-2-(4-methylphenyl)pyrimidin-5-yl]-N-methylformamido}-N-methylbutanamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
6-methyl-1-{3-oxo-3-[2-(pyrrolidine-1-carbonyl)piperazin-1-yl]propyl}-1,2-dihydropyridin-2-one
(2S,3S)-3-methyl-2-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)pentanamide
(1S,5R)-3-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-(thiophen-2-ylmethyl)-1H-pyrazole-4-carboxamide
(benzylsulfamoyl)[(2,6-difluoro-3-methoxyphenyl)methyl]amine
1-(cyclopropylmethyl)-3-hydroxy-3-(1,4-oxazepan-4-ylmethyl)piperidin-2-one
(3S,9aR)-8-(2-fluorobenzenesulfonyl)-2-methyl-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-butyl-8-{pyrazolo[1,5-a]pyridine-7-carbonyl}-2,8-diazaspiro[5.5]undecan-3-one
[(5-{1-[(4-chloro-3-fluorophenyl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
3-benzyl-4-(2,4-difluorobenzoyl)piperazin-2-one
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
methyl 3-[(2,2-dimethylpropanamido)methyl]-5-[3-(trifluoromethyl)benzenesulfonamido]benzoate
1-(4-chlorobenzoyl)-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-4-carboxamide
N-[(5-methylfuran-2-yl)methyl]-3-[1-(pyridin-2-ylmethyl)piperidin-3-yl]propanamide
3-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-N-[(4-methoxyphenyl)methyl]propanamide
1-tert-butyl-4-[3-(3-ethylphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
3-(2-chlorophenyl)-N-methyl-3-phenylpropanamide
N-(1,3-benzothiazol-2-ylmethyl)-3-(2-ethyl-5-oxopyrrolidin-2-yl)propanamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
1-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-2-(1H-pyrazol-1-yl)ethan-1-one
8-(4-methylbenzenesulfonyl)-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-(diethylamino)-3-[2-methoxy-4-({[2-(pyridin-3-yloxy)ethyl]amino}methyl)phenoxy]propan-2-ol
N-ethyl-3,3,3-trifluoro-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)propanamide
9-(2,5-dimethylfuran-3-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}benzamide
2-(4-chlorophenyl)-1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-hydroxyethan-1-one
{1-[(3-chloro-5-fluorophenyl)methyl]azepan-2-yl}methanol
2-cyclopropyl-N-({1-[(1,5-dimethyl-1H-indol-2-yl)methyl]pyrrolidin-3-yl}methyl)acetamide
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
1-(2-ethoxyethyl)-N-{[4-(hydroxymethyl)phenyl]methyl}-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
4-phenyl-5-[2-(1H-pyrazol-1-yl)ethyl]-1-[4-(pyrrolidin-1-yl)butyl]-1H-imidazole
1-[5-(azetidin-1-ylmethyl)-2-methoxyphenoxy]-3-[benzyl(methyl)amino]propan-2-ol
2-(4-amino-3-fluorophenyl)-2-(thiomorpholin-4-yl)acetic acid
2-(5-ethylpyrimidin-2-yl)-N,N-bis(propan-2-yl)benzamide
1-cyclobutanecarbonyl-N-[(1-ethyl-1H-indazol-3-yl)methyl]piperidine-4-carboxamide
3-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}isoquinoline
2-methyl-6-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}pyrimidin-4-ol
6-ethyl-2-methoxy-3-({[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
6-[4-(4-hydroxyphenyl)butan-2-yl]-1-methyl-3-phenyl-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
6-methoxy-3-[3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
3-(4-phenoxybenzoyl)-N-propylpiperidine-1-carboxamide
4-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
3-[(1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}pyrrolidin-3-yl)methyl]benzoic acid
2-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-8-fluoroquinolin-4-ol