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2-[3-methyl-1-(3-methylphenyl)-1H-1,2,4-triazol-5-yl]pyridin-4-amine
1-{2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-({4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}methyl)benzoic acid
N-(5-hydroxyadamantan-2-yl)-2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidine-1-carboxamide
N-({1-[(2E)-but-2-en-1-yl]-1,2,3,6-tetrahydropyridin-4-yl}methyl)-2-(trifluoromethyl)benzamide
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)-2-(thiophen-3-yl)acetamide
N-(3-{2-methoxy-4-[(3-methylpiperidin-1-yl)methyl]phenoxy}propyl)-2-(trifluoromethyl)benzamide
(2H-1,3-benzodioxol-5-ylmethyl)[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]methylamine
3-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]-N-cyclohexylpropanamide
(2S)-2-[(2-chloro-5-acetamidophenyl)formamido]-2-cyclopropylacetic acid
1-[(4aS,8aR)-4a-(hydroxymethyl)-6-propyl-decahydro-1,6-naphthyridin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-[4-(2-oxopyrrolidin-1-yl)phenyl]-3-[3-(1H-1,2,3-triazol-1-yl)propyl]urea
1-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
(2S)-2-amino-1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]butan-1-one
3-[1-(2H-1,3-benzodioxol-5-yl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]benzonitrile
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(5-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-{2-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
3-(2-methoxyphenoxy)-1-[1-(4-methylphenyl)cyclopropanecarbonyl]azetidine
2-{2-[(4-methylpiperazin-1-yl)methyl]phenoxy}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-(4-fluorophenyl)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)morpholine
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
N-butyl-4-oxo-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
3-(2-fluoro-4-methoxyphenyl)-4-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-1H-pyrazole
N,N-dimethyl-1-[2-methyl-5-(2-methyl-1,3-oxazol-5-yl)benzenesulfonyl]azepan-4-amine
5-chloro-2-[(1S,4S)-5-methyl-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]-3-phenyl-1H-indole
N-(2-hydroxyethyl)-3-[1-(propan-2-yl)-5-[(propan-2-yl)sulfamoyl]-1H-1,3-benzodiazol-2-yl]propanamide
4-{2-[4-(1H-pyrazol-1-yl)phenyl]pyridine-4-carbonyl}morpholine
methyl 6-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}(methyl)carbamoyl)pyridine-3-carboxylate
5-(4-cyclopentylpiperazine-1-carbonyl)-2-(4-methylphenyl)pyrimidin-4-ol
5-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
3-cyclopentyl-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
(3S,4R)-N,N-dimethyl-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-4-propylpyrrolidin-3-amine
N-(1-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
N-[(3R,4S)-1-(carbamoylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-2,6-dimethoxypyridine-3-carboxamide
N-(3,4-dimethylphenyl)-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-3-amine
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[(2S)-oxolan-2-ylmethyl]-1H-1,3-benzodiazole-5-carboxamide
(1S,5R)-6-(5-propyl-1,2-oxazole-3-carbonyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-[1-(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]oxolane-3-carboxamide
1-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-2-methyl-1,4-diazepan-5-one
(1R,5R)-6-(1H-indol-5-ylmethyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N,N-dimethyl-2-phenyl-7-[(2S)-pyrrolidine-2-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
5-methyl-1'-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[3-({[(butylcarbamoyl)methyl](methyl)carbamoyl}methoxy)phenyl]propanamide
N-(2-hydroxyethyl)-N-[(2-methoxyphenyl)methyl]-2-methyl-1-benzofuran-5-carboxamide
5-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-methylphenol
3-{1-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]piperidin-3-yl}benzoic acid
9-[2-(4-hydroxyphenyl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[3-({ethyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenyl]-3,4,5,6,7,8-hexahydroquinazolin-4-one
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2,6-dimethylquinoline-3-carboxamide