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1-cyclopropyl-N-methyl-6-oxo-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]piperidine-3-carboxamide
1-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
(4aR,7aS)-1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-[(2-cyclohexylpyrimidin-5-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
(1S,5R)-6-(cyclobutylmethyl)-3-[2-(methylsulfanyl)pyridine-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-5-phenyl-1,2-oxazole-3-carboxamide
(4aS,7aR)-1-[(4-methylphenyl)methyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3,5-dimethyl-4-{[methyl(quinolin-6-ylmethyl)amino]methyl}-1H-pyrazol-1-yl)ethan-1-ol
5-{[benzyl(methyl)amino]methyl}-N-[(2S)-1-hydroxy-3-methylbutan-2-yl]-1,2-oxazole-3-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-2-(1-methyl-3-oxopiperazin-2-yl)acetamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-5-methyl-1-phenyl-1H-pyrazole
1-[(2-benzyl-1,3-thiazol-4-yl)methyl]-3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)urea
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
1-(pyrimidin-2-yl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}piperidin-4-amine
2-ethyl-5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-4-methyl-1,3-thiazole
6-{5-[(2S)-1-methanesulfonylpyrrolidin-2-yl]-1H-1,2,4-triazol-1-yl}-2-methyl-1,3-benzothiazole
4-(2-chlorophenoxy)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine
N-{1-[4-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenyl]ethyl}acetamide
3-{[1-(6-fluoro-4-methylquinazolin-2-yl)azepan-4-yl]amino}-2,2-dimethylpropan-1-ol
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-{3-[2-(trifluoromethyl)phenyl]-1H-pyrazol-1-yl}acetamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]acetamide
1-{[4-(4-methanesulfonylphenyl)phenyl]methyl}piperidine
1-{7-[cyclohexyl(hydroxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
3-{2-[2-(3-methoxyphenyl)azetidin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
3,4-dimethyl-N-(oxolan-2-ylmethyl)-N-propyl-5-sulfamoylbenzamide
4-{2-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-2-oxoethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
1-{1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]piperidine-3-carbonyl}piperidin-4-ol
7-(1,3-benzothiazol-2-yl)-4-(quinolin-8-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-({8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)-N-methylfuran-2-carboxamide
2-amino-4-[2-(2-hydroxyethoxy)phenyl]-6-(thiophen-2-yl)pyridine-3-carbonitrile
2-(3,5-dimethylphenyl)-2-[4-(3-methoxybenzoyl)piperazin-1-yl]acetic acid
N,2,3,6-tetramethyl-N-[2-(2-oxopiperidin-1-yl)ethyl]quinoline-4-carboxamide
1-{4-[(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazin-1-yl)methyl]thiophen-2-yl}ethan-1-one
5-fluoro-2-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
methyl 2-chloro-4-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)carbamoyl}amino)benzoate
3-cyclopentyl-5-[4-(1H-pyrazol-1-yl)phenyl]-1H-1,2,4-triazole
1-(cyclohexylmethyl)-N,N-dimethyl-5-{methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(benzylsulfamoyl)({[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl})amine
2-{4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-ethyl-1,2-oxazole-4-carboxamide
1-[3-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(thiophen-2-yl)propan-1-one
(4aS,7aR)-1-[2-(2-methoxyphenyl)acetyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,5R)-1-[(3,4-dimethoxyphenyl)methyl]-N3-[(3,5-dimethylphenyl)methyl]-N5-(4-fluorophenyl)piperidine-3,5-dicarboxamide
2-methyl-1-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-1,4-diazepan-5-one
(2S,4S)-4-amino-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-fluoro-4-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)pyridine
5-(4-chloro-2-methoxyphenoxymethyl)-N-(oxan-4-ylmethyl)-1,2-oxazole-3-carboxamide
2-{2-[methyl(phenyl)amino]acetyl}-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
4-{4-[butyl(methyl)amino]piperidin-1-yl}-N-(1-phenylethyl)benzamide