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(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-1-[(3,4-dimethoxyphenyl)methyl]-N-(2-methylpropyl)piperidine-3-carboxamide
N-[(2,5-dimethylphenyl)methyl]-3-[(4-fluorophenyl)formamido]propanamide
N-(2-methoxyethyl)-2-methyl-3-({[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]carbamoyl}amino)benzamide
5-(5-methoxyfuran-2-yl)-1-[(3-methylphenyl)methyl]-1H-1,2,4-triazole
3-benzyl-8-[(4-methoxyphenyl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]-1-methylimidazolidin-2-one
(4aS,8aR)-6-(2-aminopyrimidin-4-yl)-1-methanesulfonyl-decahydro-1,6-naphthyridine-4a-carboxylic acid
3-[2-(4-fluorophenyl)ethyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperidine
2-amino-4-(3-ethoxy-4-hydroxyphenyl)-6-(3-fluorophenyl)pyridine-3-carbonitrile
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-hydroxy-3-methoxybenzamide
(2,3-dihydro-1-benzofuran-2-ylmethyl)({[5-(furan-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl})methylamine
5-[4-(benzyloxy)piperidine-1-carbonyl]-4-ethyl-1,3-thiazol-2-amine
{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(1H-pyrazol-3-ylmethyl)amine
2-{3-[3-(morpholin-4-ylmethyl)phenyl]phenoxy}propanamide
[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl][1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amine
5-{2-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
methyl 6-({[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]carbamoyl}amino)-1,2,3,4-tetrahydroquinoline-1-carboxylate
2-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-6-methylpyridine-3-carboxylic acid
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
N-[1-(furan-2-ylmethyl)piperidin-4-yl]-2-(methylamino)pyridine-4-carboxamide
1-benzyl-4-oxo-N3-(3-phenylpropyl)-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-(2-methylpropyl)-3-{2-oxo-2-[4-(pyrazin-2-yl)piperazin-1-yl]ethyl}piperazin-2-one
methyl 2-[8-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
3-(4-chloro-1H-pyrazol-1-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)propanamide
methyl 5-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2-acetyl-8-[(dimethyl-4H-1,2,4-triazol-3-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]pyrrolidin-3-yl}benzoic acid
4-{3-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]phenyl}phenol
8-[2-(4-fluorophenoxy)acetyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[4-(4-fluorophenyl)oxane-4-carbonyl]-3-(1H-pyrazol-5-yl)piperidine
3-(4-benzyl-1H-pyrazol-5-yl)-1-(dimethyl-1,2-oxazole-4-carbonyl)piperidine
5-({5-[(2E)-but-2-en-2-yl]-4-phenyl-1H-imidazol-1-yl}(cyclopropyl)methyl)-1-methyl-1H-1,2,4-triazole
3-{[2-hydroxy-3-(3-methoxyphenoxy)propyl]amino}butan-1-ol
1-methanesulfonyl-4-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]-1,4-diazepane
{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
3-phenyl-1-[1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]propan-1-one
(1R,5S)-N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-6-azabicyclo[3.2.1]octane-6-carboxamide
1-{2-methylthieno[2,3-d]pyrimidin-4-yl}-N-[3-(pyridin-4-yl)propyl]piperidin-4-amine
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
({6-[(3-fluorophenyl)methoxy]-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl}methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
2-(5-fluoro-2-methylphenyl)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-[5-(2,4,6-trimethylphenyl)pyridin-2-yl]acetamide
3-[(2R,3R,6R)-5-[(3-fluorophenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
1-(7-{[(2S)-4-methyl-2-phenylpiperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
(1R,7S)-N-methyl-3-[(3-methylphenyl)methyl]-4-oxo-N-[2-(pyridin-2-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-[(4-formyl-1,4-diazepan-1-yl)methyl]-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
3-acetamido-N-[(2-phenoxypyridin-3-yl)methyl]benzamide
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-(naphthalen-1-ylmethyl)-1,2-oxazole-3-carboxamide
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide