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(3S)-3-(3-methoxyphenyl)-1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidine
6-methoxy-3-({4-[(2-methylphenyl)methyl]piperazin-1-yl}methyl)-1H-indazole
11-[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
2-[4-(1H-indol-3-ylmethyl)-1-(3-methylbutyl)piperazin-2-yl]ethan-1-ol
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-3-(3-methylpiperidin-1-yl)propan-1-one
2-amino-6-(4-hydroxyphenyl)-5-methyl-4-(piperidin-4-yl)pyridine-3-carbonitrile
(1S,5R)-3-{[2-(4-fluorophenyl)imidazo[1,2-a]pyridin-3-yl]methyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonane
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carboxamide
1-[(4-methylphenyl)methyl]-3-[1-(2-phenylethyl)piperidin-3-yl]urea
(3S,4R)-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-(2-hydroxypropanoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N,N-diethyl-7-methoxy-2-[2-(methylamino)pyrimidin-5-yl]quinoline-4-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}acetamide
3-ethyl-N-[4-(2-fluorophenoxy)phenyl]-3-(hydroxymethyl)piperidine-1-carboxamide
1-{[3-(difluoromethoxy)phenyl]methyl}-3-[4-methyl-3-(2-oxopyrrolidin-1-yl)phenyl]urea
1-[4-({[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]imidazolidin-2-one
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
3-chloro-5-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2-dihydropyridin-2-one
2-(2-chloro-6-fluorophenyl)-2-[4-(morpholin-4-yl)piperidin-1-yl]acetic acid
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(3-chloro-1H-1,2,4-triazol-5-yl)propan-1-one
5-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-N-ethyl-4-methyl-1,3-thiazol-2-amine
1-{2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl}-4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine
N-(3-ethoxypropyl)-1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(4aS,8aR)-1-[(2-aminopyridin-3-yl)methyl]-6-(pyrazin-2-yl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
7-(oxan-4-yl)-2-[2-(4H-1,2,4-triazol-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
8-[2-(azepan-1-yl)acetyl]-2-benzyl-2,8-diazaspiro[4.5]decan-3-one
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
6-(1-methyl-1H-imidazol-2-yl)-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)pyridazin-3-amine
5-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1-ethyl-1H-indole
N-[(2,3-dimethoxyphenyl)methyl]-4-hydroxy-2-phenylpyrimidine-5-carboxamide
(1R,2R,6S,7S)-4-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4-azatricyclo[5.2.1.02,6]decane
1-(3-{[3-(pyrrolidine-1-carbonyl)-1,2-oxazol-5-yl]methoxy}phenyl)ethan-1-one
2-(morpholin-4-ylmethyl)-4-[4-(pyridin-3-yl)pyrimidin-2-yl]-1,4-oxazepane
4-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}benzoic acid
4-({[(3-hydroxypyrrolidin-3-yl)methyl]amino}methyl)-N,N-dimethylbenzene-1-sulfonamide
N-[2-(3-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]-2-(thiophen-3-yl)acetamide
2-[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)pyrrolidin-2-yl]pyridine
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-(piperidine-1-carbonyl)pyridine
2,6-dimethyl-3-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
2-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-N-(pyridin-2-ylmethyl)acetamide
methyl (2S,4S,5R)-1,2-dimethyl-4-{methyl[2-(pyridin-2-yl)ethyl]carbamoyl}-5-phenylpyrrolidine-2-carboxylate
2-{4-[1-(3-methoxyphenyl)piperidin-4-yl]-1-methylpiperazin-2-yl}ethan-1-ol
4-(azepan-1-yl)-5-methyl-N-[2-(thiophen-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
2-(adamantan-1-ylsulfanyl)-N-[1-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]acetamide
N-[2-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)quinolin-6-yl]acetamide
1-(2-methoxyethyl)-3-(5-methyl-2,1,3-benzothiadiazol-4-yl)-1-(thiophen-2-ylmethyl)urea
8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[1-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]benzoic acid
1-{3-[2-(4-chlorophenyl)morpholin-4-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one