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1-(3-{4-[2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidine-1-carbonyl}phenyl)pyrrolidin-2-one
ethyl[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
2-(2-{[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}phenyl)-3H,4H,5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-one
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-(cyclohexylmethyl)-N-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
2-[4-(2-methyl-1-benzofuran-5-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
N-ethyl-2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]acetamide
2-({[(3R,4R)-1-[(4-fluorophenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[(3S,4R)-1-(4-chloro-3-fluorobenzoyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(4-methylphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N3-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2,2-dimethyloxane-4-carboxamide
phenyl(1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-yl)methanol
2-methyl-6-[2-(1,2,5-thiadiazole-3-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
(3R,4S)-4-cyclopropyl-1-{4-[(2-fluorophenyl)methoxy]benzoyl}pyrrolidin-3-amine
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyridin-3-ylmethyl)acetamide
(2R)-2-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-3-hydroxypropanoic acid
4-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-2-phenylmorpholine
2-[4-(2,5-dimethoxyphenyl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-1,2,3-triazol-4-yl)acetamide
4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]morpholine-2-carboxamide
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-1-phenyl-1H-1,2,3-triazole-4-carboxamide
4-[3-(thiomorpholine-4-carbonyl)benzenesulfonyl]-1,4-oxazepane
N-[2-methyl-2-(morpholin-4-yl)propyl]-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1-(6-methyl-2H-1,3-benzodioxol-5-yl)urea
1'-benzoyl-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(2-chloro-4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}phenoxy)propanoic acid
(4aS,8aR)-1-(3-aminopropyl)-6-[3-(thiophen-3-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,3-benzodiazole
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
1-[2-(dimethylamino)acetyl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
(3S,4S)-1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-4-propylpyrrolidine-3-carboxylic acid
1-{1-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]piperidin-4-yl}-2-phenylethan-1-ol
1-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-[(1-ethyl-1H-indol-6-yl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
3-(2-phenylethyl)-5-[(2,2,2-trifluoro-1-phenylethoxy)methyl]-1H-1,2,4-triazole
4-[(3,4-dimethoxyphenyl)methyl]-3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]piperazin-2-one
1-cyclopentanecarbonyl-N-[(5-ethylpyridin-2-yl)methyl]-N-methylpiperidine-4-carboxamide
4-{2-[1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]ethyl}phenol
1-[(2-chlorophenyl)methyl]-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-(2-hydroxyethyl)-8-[2-(3-methylphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-cyclopropyl-N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-5-oxopyrrolidine-3-carboxamide
1-cyclopentyl-3-(piperidine-1-carbonyl)-5-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1,4-dihydropyridin-4-one
1-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carbonyl)piperidin-4-ol
5-methyl-1'-[4-(trifluoromethyl)benzoyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
8-methoxy-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
(1R,2S)-1-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-2,3-dihydro-1H-inden-2-ol
2,5-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(pyridin-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
{1-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-propylpiperidin-3-yl}methanol