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5-({[1-(6-chloro-1,3-benzothiazol-2-yl)piperidin-4-yl](methyl)amino}methyl)pyrimidin-2-amine
2-({[1-butyl-2-(cyclohexanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)amino)-1-phenylethan-1-ol
4-[5-(methoxymethyl)furan-2-carbonyl]-2-(3-phenylpropyl)morpholine
2-cyclopropyl-4-phenyl-9-(1H-pyrrole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[3-cyclopentyl-1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}ethan-1-one
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-4-oxo-4-phenylbutanamide
5-amino-N-(2,2-dimethyloxan-4-yl)-2-(2-methoxyphenyl)-1-methyl-1H-1,3-benzodiazole-7-carboxamide
2-[3-(3-methoxyphenoxymethyl)-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl]-6-methylpyridine
1-(4-benzyl-6-hydroxy-1,4-diazepane-1-carbonyl)cyclopropane-1-carboxamide
1-(2-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}phenyl)ethan-1-one
6-{4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-methyl-4-sulfamoyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)benzamide
2-(dimethyl-1,3-thiazol-5-yl)-N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]acetamide
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-methylacetamide
1-(2-cyclohexylethyl)-3-[(cyclopentylamino)methyl]-3-hydroxypiperidin-2-one
4-(1H-imidazol-1-ylmethyl)-2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazole
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(3-methylpyrazin-2-yl)pyrrolidin-3-yl]methanol
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-4-(piperidin-1-ylmethyl)benzamide
2-(4-chlorophenyl)-5-(3,4-difluorobenzoyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-{3-[2-(1-benzofuran-2-yl)-1H-imidazol-1-yl]propyl}piperidin-3-ol
4-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carbonyl)piperazin-2-one
(3aR,6aR)-2-(3-ethoxypropanoyl)-5-(1H-imidazol-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
9-(2,6-dimethylpyrimidine-4-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-1,3-benzoxazol-2-amine
N-cyclopropyl-2-[4-(2-methoxyphenoxy)piperidin-1-yl]pyridine-4-carboxamide
4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)-1-[(5-methylfuran-2-yl)methyl]piperidine
2-cyclopropyl-8-[4-(trifluoromethyl)pyridin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
(2S,4R)-4-amino-1-[(2-methoxypyrimidin-5-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-(4-{[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}piperidin-1-yl)-N-(1-phenylethyl)benzamide
2-[9-(2-amino-6-methylpyrimidin-4-yl)-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]acetamide
1-[4-(morpholine-4-carbonyl)phenyl]-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]piperidin-4-amine
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}(ethyl)(pyridin-4-ylmethyl)amine
3-[4-(1-hydroxy-3-methylbutyl)piperidine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
2-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)benzonitrile
2-({[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)amino)-N,N-dimethylpropanamide
N,N-dimethyl-6-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]pyrazin-2-amine
N,N-diethyl-1-[2-(morpholin-4-yl)-6-phenylpyridine-3-carbonyl]piperidine-3-carboxamide
(2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-(5,6,7,8-tetrahydro-1,6-naphthyridine-6-carbonyl)pyrrolidine-2-carboxylic acid
3-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-1-(2-phenylethyl)urea
2-methyl-4-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-1,2-dihydrophthalazin-1-one
2-(3-{3-[2-(pyridin-3-yl)-1,3-benzoxazol-5-yl]phenyl}-1H-pyrazol-1-yl)acetamide
1-(benzyloxy)-8-[5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carbonyl]-1,8-diazaspiro[4.5]decan-2-one
2-(2-hydroxyphenoxy)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
3-(3,4-difluorophenyl)-5-(3-methylthiophene-2-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-(1-methyl-1H-imidazole-5-carbonyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
9-[(2S)-2-hydroxy-3-phenylpropanoyl]-2,9-diazaspiro[5.5]undecan-3-one
6-[4-(4-methoxypyrimidin-2-yl)piperazine-1-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
(3S,4R)-1-[3-(cyclopentylcarbamoyl)propanoyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-2-(3,4,5-trimethoxyphenyl)pyridine
methyl 5-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}-2-hydroxybenzoate