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8-[3-(3-fluorophenoxymethyl)piperidine-1-carbonyl]quinoline
1-{4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}pyrrolidin-3-amine
2-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)-4,5,6,7-tetrahydro-1,3-benzothiazole
5-acetyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-{4-[3-(trifluoromethyl)phenoxy]piperidine-1-carbonyl}pyridine
3-(1H-imidazol-1-yl)-1-[4-(3-methoxybenzoyl)piperazin-1-yl]butan-1-one
(2R,6S)-4-(1-{1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}piperidin-4-yl)-2,6-dimethylmorpholine
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1-cyclopropyl-5-oxopyrrolidine-3-carboxamide
2-tert-butyl-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-4-hydroxypyrimidine-5-carboxamide
4-(3-{3-[3-(3-chloropyridin-2-yl)phenyl]-1H-pyrazol-1-yl}propyl)morpholine
1-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylamino)ethan-1-one
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-hydroxyacetamide
N-(cyclopropylmethyl)-N-(2-methoxyethyl)-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
N-[2-(azepan-1-yl)-2-phenylethyl]-1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-(2,3-dimethylphenyl)-4-[4-(piperidin-3-yl)benzoyl]piperazine
1-(2-methylphenyl)-4-{1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidin-3-yl}piperazine
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{[3-(trifluoromethoxy)phenyl]methyl}acetamide
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
N-methyl-6-oxo-1-[2-(pyridin-2-yl)ethyl]-N-(thiophen-3-ylmethyl)piperidine-3-carboxamide
8-fluoro-3-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
N-{3-[ethyl(phenyl)carbamoyl]phenyl}-2-methoxypyridine-3-carboxamide
4-{1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]azetidin-3-yl}morpholine
3-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-1-[1-(1H-indol-2-yl)ethyl]-1-methylurea
1-(4-{[(7-methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)amino]methyl}piperidin-1-yl)-2-methylpropan-1-one
4-(hydroxymethyl)-1-[6-(trifluoromethyl)pyridin-2-yl]piperidin-4-ol
N-(furan-2-ylmethyl)-2-{3-[3-(1-methyl-1H-pyrazol-4-yl)phenyl]-1H-pyrazol-1-yl}acetamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-2-methoxy-N-(oxolan-2-ylmethyl)benzamide
3-cyclopropaneamido-N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N,4-dimethylbenzamide
butyl 2-(1,3-benzothiazol-2-yl)pyrrolidine-1-carboxylate
3-{[(1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
2-{[3-(azepane-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-yl](methyl)amino}ethan-1-ol
2-[benzyl(methyl)amino]-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
9-(azepane-4-carbonyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-[3-fluoro-5-(2-methylpropoxy)phenyl]-6-(pyrrolidine-1-carbonyl)pyrazine
methyl 2-{[(3-fluorophenyl)methyl]sulfamoyl}-6-(pent-4-enoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
N-(cyclohexylmethyl)-1-cyclopropyl-4-oxo-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
N-[2-(4-phenyl-1H-imidazol-5-yl)quinolin-6-yl]acetamide
(3S,4R)-4-(pyridin-4-yl)-1-(quinoline-2-carbonyl)pyrrolidine-3-carboxylic acid
(1R,2R,6S,7S)-4-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
4-phenyl-N-{[1-(pyrimidin-2-ylmethyl)piperidin-3-yl]methyl}benzamide
[(3-methylpyridin-2-yl)methyl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)(propan-2-yl)amine
methyl[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl][(2E)-2-methylbut-2-en-1-yl]amine
1-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-3-ol
2-(3,4-dimethoxyphenyl)-8-methyl-3-(1,4-oxazepan-4-ylmethyl)quinoline
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-(morpholin-4-yl)ethan-1-one
2-amino-N-[3-(1H-indol-1-yl)propyl]-4-methylpyrimidine-5-carboxamide
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-(2-hydroxyethyl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]urea
(3R,9R)-11-benzoyl-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione