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1-{5-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]thiophen-2-yl}ethan-1-one
3-methyl-5-({2-[4-(propan-2-yl)-1,3-thiazol-2-yl]-1H-imidazol-1-yl}methyl)-1,2-oxazole
3-cyclopentyl-N-{2-[4-(4-methyl-1,4-diazepane-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}propanamide
5-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-3-(5-methylfuran-2-yl)-1H-pyrazole
(3S,4R)-1-(1H-indole-3-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(4-methylpyrimidine-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[(2-methylphenyl)methyl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
(2S,4R)-N-ethyl-4-[2-(pyridin-3-yl)acetamido]-1-(thiophen-2-ylmethyl)pyrrolidine-2-carboxamide
(2R)-2-acetamido-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]propanamide
1-(5-tert-butyl-2-methoxyphenyl)-3-[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]urea
3-(2-ethyl-4-methyl-1H-imidazol-1-yl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
6-[2-(1H-imidazol-4-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
{[5-(2-chlorophenyl)furan-2-yl]methyl}(methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
2-methyl-9-({2-[(oxolan-2-ylmethyl)amino]pyrimidin-5-yl}methyl)-2,9-diazaspiro[5.5]undecan-3-one
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl][(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)amine
(4aR,7aS)-1-(1H-imidazol-4-ylmethyl)-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(2-chloro-4,6-dimethoxyphenyl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
{5-[(3R,4S)-3-amino-4-phenylpyrrolidine-1-carbonyl]-1H-1,3-benzodiazol-2-yl}methanol
3-cyclopentyl-1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-[(4-methoxyphenyl)methyl]pyrrolidine-1-carboxamide
2-[4-(cyclohexylmethyl)-1-[(3,5-dimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,4-dioxane-2-carboxamide
N-[(3S,4R)-1-(6,8-dimethoxy-4-methylquinolin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
2-methoxy-1-{1'-[2-(4-methylphenyl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
(1R,5R)-6-(1,3-dimethyl-1H-indole-2-carbonyl)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
1-[4-({3-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)thiophen-2-yl]ethan-1-one
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-[(2-methylpyrimidin-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1H-indole-6-carboxamide
5-cyclobutanecarbonyl-1'-(1-methyl-1H-imidazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(2-methoxyacetyl)-N-[(3-phenylphenyl)methyl]piperidine-3-carboxamide
1-(azocan-1-yl)-3-[2-methoxy-5-({[3-(pyridin-3-yl)propyl]amino}methyl)phenoxy]propan-2-ol
3-amino-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}butan-1-one
5-methyl-3-(4-{[4-(5-methylfuran-2-yl)-1H-1,2,3-triazol-1-yl]methyl}phenyl)-1,2,4-oxadiazole
2-[4-(1,3-oxazol-5-yl)benzoyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
N-methyl-5-phenyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-oxazole-3-carboxamide
3-(4-chlorophenyl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-3-phenylpropanamide
{[5-(1-{imidazo[1,2-a]pyridine-3-carbonyl}piperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
N-(3-methyl-1,2,4-thiadiazol-5-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
3-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-5,6-dimethyl-1,2-dihydropyridin-2-one
4-[5-(ethoxymethyl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]-3-methylpyridine
1-[2-methoxy-5-({[2-(1,3-thiazol-4-yl)ethyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
2-cyclopropyl-6-oxo-N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]-1,6-dihydropyrimidine-5-carboxamide
2-(4-methyl-6-{4-[(oxolan-2-ylmethyl)amino]piperidin-1-yl}pyrimidin-2-yl)phenol
2-ethoxy-5-(2-{[2-(pyridin-4-yl)ethyl]amino}pyrimidin-4-yl)benzoic acid
2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-4-carbonitrile
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-propylpyridine-4-carboxamide
2-acetyl-8-[(2-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2,6-difluoro-N-{2-[1-(3-fluoropropyl)-1,2,5,6-tetrahydropyridin-3-yl]ethyl}benzamide
2-(5-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)phenol
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-methylpiperidine