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6-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]pyridine-2-carboxylic acid
1-[2-({[2-(2-hydroxyethoxy)phenyl]methyl}(methyl)amino)ethyl]cyclopentan-1-ol
5-[4-(aminomethyl)piperidin-1-yl]-2-(pyrimidin-2-ylmethyl)-2,3-dihydropyridazin-3-one
N-cyclopentyl-4-oxo-4-[4-(2-propoxyethyl)piperazin-1-yl]butanamide
4-[2-(4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-1-yl)ethyl]morpholine
(3aR,6aS)-2-ethyl-1-oxo-5-(thiophene-2-sulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 3-{[(2-cyclopropylquinolin-4-yl)formamido]methyl}-5-(furan-3-amido)benzoate
2-(1-methyl-1H-pyrazole-4-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
{1-[(3-chloro-1H-indol-2-yl)methyl]-3-methylpiperidin-3-yl}methanol
2-(4-fluorophenoxymethyl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
2-(2,3-dihydro-1-benzofuran-7-yl)-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]acetic acid
1-[4-(4-{[(2,3-difluorophenyl)methyl]amino}piperidin-1-yl)benzoyl]piperidin-3-ol
5-({2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}methyl)-2,1,3-benzoxadiazole
2-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-3-methylpyrazine
(3aR,6aR)-2-[(3-hydroxyphenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3aS,6aS)-5-{[3-(furan-2-yl)phenyl]methyl}-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{2-oxo-1-oxa-3,7-diazaspiro[4.5]decane-7-carbonyl}thiophene-3-sulfonamide
4-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-6-(methoxymethyl)pyrimidine
N3,N3-dimethyl-N5-(2-methylquinolin-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3,5-dicarboxamide
N-[1-(4-fluorophenyl)-2-methylpropan-2-yl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
8-[(3-hydroxyphenyl)methyl]-1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]acetamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
2-methoxy-1-[1'-(2-methoxypyridine-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-(3,5-dimethoxyphenyl)-3-{1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}propanamide
ethyl 2-{[2-({[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}carbamoyl)phenyl]amino}acetate
5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-ethyl-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1,2-oxazole-3-carboxamide
N-(pyrimidin-4-ylmethyl)-3-[(2,2,2-trifluoroethyl)sulfamoyl]benzamide
5-(1-carboxycyclopropanecarbonyl)-1-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-methyl-5-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
N-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methoxybenzamide
5-({3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1-ethyl-1H-1,2,4-triazole
3,3-dimethyl-N-[(3-methyl-1H-pyrazol-5-yl)methyl]-2-methylidenebicyclo[2.2.1]heptane-1-carboxamide
1-(4-{5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)-2,2-dimethylpropan-1-one
4-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-1λ6-thiane-1,1-dione
(3R,4R)-1-(4-amino-6,7-dimethoxyquinazolin-2-yl)-4-ethylpiperidine-3,4-diol
N-ethyl-N-[2-(4-methylbenzenesulfonyl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-(cyclohexylmethyl)-6-oxo-N-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidine-3-carboxamide
5-[3-carboxy-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid
({4-cyclopropyl-5-[1-(pyridine-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1H-indol-5-ylmethyl)piperidin-3-ol
N-[(1-hydroxycyclohexyl)methyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
1-(2-{4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}ethyl)piperidine-4-carboxamide
N-[2-(4-fluorophenyl)ethyl]-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-2,2-dimethyloxane-4-carboxamide
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)-2-(trifluoromethyl)benzamide
7-(cyclohexylmethyl)-2-(furan-2-carbonyl)-2,7-diazaspiro[4.5]decane
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(prop-2-en-1-yl)(pyridin-2-ylmethyl)amine
1-methyl-4-(quinolin-2-yl)-1,4-diazepan-6-ol
(2S,4S)-4-amino-N-(2H-1,3-benzodioxol-5-ylmethyl)-1-methyl-N-(pentan-3-yl)pyrrolidine-2-carboxamide