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N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-2-(thiophen-3-yl)acetamide
6-{3-oxo-3-[3-(phenylamino)piperidin-1-yl]propyl}-2,3,4,5-tetrahydropyridazin-3-one
1-(3-phenyl-1,2-oxazole-4-carbonyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
N-(adamantan-1-yl)-N'-ethyl-N'-(pyridin-4-ylmethyl)propanediamide
4-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-1-methyl-3-(propan-2-yl)piperazin-2-one
(1S,4S)-2-(1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carbonyl)-2-azabicyclo[2.2.1]heptane
ethyl[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](1H-indol-7-ylmethyl)amine
(3S,7S)-5-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
2-(4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-1-(3-phenylpropyl)piperazin-2-yl)ethan-1-ol
2-methyl-4-(4-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}phenyl)butan-2-ol
2-ethoxy-4-[1-(propan-2-yl)-1H-imidazol-2-yl]phenol
1-[(4-ethylphenyl)methyl]-5-oxo-N-[2-(pyrazin-2-yl)ethyl]pyrrolidine-3-carboxamide
7-(1,3-benzothiazol-2-yl)-4-(2-hydroxyethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-(2-phenylbenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
N-[4-(furan-2-yl)butan-2-yl]pyrazolo[1,5-a]pyridine-7-carboxamide
6-[3-(3-hydroxy-3-methylbutyl)benzoyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
2-amino-6-(3-fluorophenyl)-4-[2-(furan-2-yl)pyrimidin-5-yl]pyridine-3-carbonitrile
N-[(1-cyclohexylpiperidin-3-yl)methyl]-2-(2-methoxyphenoxy)acetamide
4-hydroxy-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
1-(3-methanesulfonamido-4-methoxyphenyl)-3-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]urea
2-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1,3-oxazole-4-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-2-(methylamino)acetamide
1-benzyl-N,N-dimethyl-5-(4-methylpiperidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(4-phenyl-1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-imidazol-5-yl)benzonitrile
N-({7-[2-(2-methoxyphenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-3-yl)acetamide
2-hydroxy-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methylpentanamide
3-methyl-N-{1-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
3-benzyl-1-(3-methoxypropyl)-8-[(1-methyl-1H-indol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(pyrazin-2-yl)acetamide
1-cyclohexyl-4-[3-(2-phenylpropyl)-1,2-oxazole-5-carbonyl]piperazin-2-one
4-[(2,6-dimethylpyridin-3-yl)oxy]-1-(4-methoxypyrimidin-2-yl)piperidine-4-carboxylic acid
N-[(3-chlorophenyl)methyl]-N-propylfuran-3-carboxamide
ethyl 3-[(2-methylphenyl)methyl]-1-(pyridin-4-ylmethyl)piperidine-3-carboxylate
2-{2-[2-amino-3-cyano-6-(furan-2-yl)pyridin-4-yl]-6-methoxyphenoxy}propanoic acid
1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(3-methoxyphenyl)piperidine
2-(3-methoxypropyl)-9-[(2E)-3-phenylprop-2-en-1-yl]-2,9-diazaspiro[5.5]undecan-3-one
4-(4-fluorophenyl)-4-oxo-N-(quinolin-2-ylmethyl)butanamide
2-(2,4-difluorophenoxy)-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}acetamide
2-[4-(1-benzofuran-2-ylmethyl)-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
4-{[3-(4,6-dimethylpyridin-2-yl)phenyl]methyl}morpholine
2-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carbonitrile
8-methyl-3-{[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]methyl}-2-(thiophen-2-yl)quinoline
1,6-dimethyl-N-[(5-methyl-1H-imidazol-4-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
[(3S,5R)-1-[2-(benzyloxy)benzoyl]-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
methyl (2R,4S)-1-[(2,3-dimethoxyphenyl)methyl]-4-hydroxypiperidine-2-carboxylate
(1R,5R)-6-benzyl-3-(4-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
N,15-dimethyl-N-(2-methylpropyl)-13-oxo-9-(pyridin-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
2-[N-(4-methylphenyl)methanesulfonamido]-N-[3-(oxolan-3-yl)propyl]acetamide