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(2S)-N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-1-(piperidin-4-yl)pyrrolidine-2-carboxamide
2-(1,3-benzoxazol-2-yl)-1-[4-(pyridin-3-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
3-(1H-1,2,3-benzotriazol-1-yl)-1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]propan-1-one
8-[(2-fluoro-4-methylphenyl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[5-(ethylsulfanyl)-1,3,4-thiadiazol-2-yl]-2-[(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)amino]acetamide
4-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-2-[(4-methoxyphenyl)methyl]morpholine
4-({2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}amino)-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
N-[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
4-[4-(pyridin-2-yl)butyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
5-ethyl-N-(morpholin-2-ylmethyl)-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
(1S,5R)-3-(ethanesulfonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1R,5R)-6-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-methyl-7-(methylsulfanyl)-2-[4-(morpholin-4-ylmethyl)piperidin-1-yl]quinoline
(1R,2S)-N-(prop-2-en-1-yl)-2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}cyclohexane-1-carboxamide
(3aR,6aR)-2-(cyclopentylcarbamoyl)-5-(pyridin-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(2-fluorophenyl)methyl]-4-methyl-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
1-[1-(3-methylbutyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-{5-[(benzylsulfamoyl)amino]-2-methoxyphenyl}methanesulfonamide
N-[(8-methoxyquinolin-2-yl)methyl]-N-methylthian-4-amine
N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(furan-2-carbonyl)-4-(5-phenyl-1,2-oxazole-4-carbonyl)-1,4-diazepane
5-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
8-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
2-{[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)amino}pyridine-4-carbonitrile
2-[5-oxo-3-phenyl-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-2-[4-(dimethylamino)phenyl]ethan-1-one
(3S,4R)-4-(4-fluorophenyl)-1-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]pyrrolidine-3-carboxylic acid
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]but-3-enamide
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-(morpholin-4-yl)pyrimidine-5-carboxamide
1-[(2-fluoro-4-methoxyphenyl)methyl]-4-[(3-fluorophenyl)methyl]-1,4-diazepan-5-one
3-{[1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1H-1,2,3-triazol-4-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
8-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1H-pyrazole-3-carbonyl]-2-methyl-2,8-diazaspiro[4.5]decane
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N,N-dimethylacetamide
2-(3-hydroxypyridine-2-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
(2R)-2-hydroxy-1-[7-(1,2,3,4-tetrahydroquinoline-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]propan-1-one
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2-(pyridin-3-yl)acetamide
(3S,4R)-4-(pyridin-4-yl)-1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]pyrrolidine-3-carboxylic acid
4-chloro-1-methyl-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
3-ethyl-N-[1-(2-methylphenoxy)propan-2-yl]-1H-pyrazole-4-carboxamide
N-{3-[(trifluoromethyl)sulfanyl]phenyl}-2,8-diazaspiro[4.5]decane-2-carboxamide
2-(oxolan-2-ylmethyl)-9-(pyrrolidine-1-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{2-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethyl}-1H-indole
2-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetamide
2-(2H-1,3-benzodioxol-5-yl)-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)acetamide
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1H-imidazol-2-yl)benzamide
8-[(4-methanesulfonylphenyl)methyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
(1S,4R)-1-[({4-[2-(cyclopentylmethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}sulfonyl)methyl]-7,7-dimethylbicyclo[2.2.1]heptan-2-one
N-butyl-N-methyl-3-({methyl[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
(4aS,8aR)-1-[2-(pyridin-2-yl)ethyl]-6-(thiophen-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1,3-benzothiazole