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N-{3H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N,4,6-trimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3,5-dimethyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-ethyl-1H-pyrazole-4-carboxamide
3-[(3R,4S)-1-[2-(methylamino)pyridine-4-carbonyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-[(2-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)acetamide
3-(3-hydroxyquinoxalin-2-yl)-N-(1,3-thiazol-2-ylmethyl)propanamide
N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)-2-(pyridin-4-yl)acetamide
5-tert-butyl-N-(2,3-dihydro-1-benzofuran-3-yl)-1,3,4-oxadiazol-2-amine
N-[2-(pyridin-2-ylmethoxy)phenyl]oxan-4-amine
5-methyl-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-1,2-oxazole-4-carboxamide
N-[(2-fluorophenyl)methyl]-5-[(2-hydroxyethyl)(methyl)amino]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
[(3S,5R)-1-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
4-(2H-1,3-benzodioxol-5-yl)-3-[2-(phenylamino)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-methyl-7-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-3,4-dihydroquinazolin-4-one
(4aR,7aS)-1-acetyl-4-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2,6-dimethyl-4-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]quinoline
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-(dimethylamino)-2,3-dihydro-1H-indene-2-carboxamide
N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
N-methyl-N-[2-({10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)ethyl]methanesulfonamide
1-[4-({[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl](methyl)amino}methyl)thiophen-2-yl]ethan-1-one
1-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]-2-(pyridin-3-yloxy)ethan-1-one
1-(4-methanesulfonamido-3-methylphenyl)-5-oxopyrrolidine-3-carboxylic acid
8-(3-hydroxy-2-methylbenzoyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(cyclopropylmethyl)-3-hydroxy-3-{[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]methyl}piperidin-2-one
3-(1H-1,2,3-benzotriazol-4-yl)-1-{1-[(4-fluorophenyl)methyl]piperidin-3-yl}urea
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-3-(3-methoxypropyl)piperidine
(3S,4S)-4-(dimethylamino)-1-[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidin-3-ol
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-ethoxyethan-1-one
N-(2-{7-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2,4-dimethylbenzamide
3-{4-[(3-cyanophenyl)methyl]piperazine-1-carbonyl}piperidine-1-carboxamide
(1R,2R,6S,7S)-4-(9H-purin-6-yl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
1-{3-[(dimethylsulfamoyl)amino]phenyl}-3-[3-(4H-1,2,4-triazol-4-yl)propyl]urea
N-[3-(dimethylcarbamoyl)-5-[({1-[3-(trifluoromethyl)phenyl]propan-2-yl}amino)methyl]phenyl]pyridine-2-carboxamide
N-[3-(3-ethylphenoxy)propyl]-3-hydroxy-N-methylpyridine-2-carboxamide
4-chloro-N-(2-{[(3-hydroxypiperidin-3-yl)methyl]amino}ethyl)benzene-1-sulfonamide
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(5-methylpyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(ethylamino)-N-(furan-3-ylmethyl)-N-methylpyrimidine-5-carboxamide
1-{[2-(4-chlorophenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-1,4-diazepan-5-one
4-(2,6-dimethylpyridin-3-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}pyrimidin-2-amine
1-[2-(naphthalen-2-yloxy)propanamido]cyclohexane-1-carboxamide
N-[2-(pyrazin-2-yl)ethyl]-1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]piperidin-4-amine
(4-methyl-5-{1-[(3-methylquinoxalin-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methanol
4-[1-(2H-1,3-benzodioxol-5-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-6-methyl-1,2-dihydroquinolin-2-one
8-(3-chloro-4-fluorobenzoyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(4-{[(2S)-3-methylbutan-2-yl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
1-(2-fluoro-5-methylbenzenesulfonyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
N-[(4-fluorophenyl)methyl]-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-(prop-2-en-1-yl)acetamide
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N,N-dimethylpiperidine-1-carboxamide