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4-methyl-6-{3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl}-1,3-benzothiazol-2-amine
N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-{3-oxo-3-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]propyl}-1,2-dihydropyridin-2-one
(3aR,6aS)-5-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2,3-dimethylphenyl)-N-({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-{[6-chloro-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-4-ethylbenzene-1-sulfonamide
N-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
4-ethyl-5-methyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]thiophene-3-carboxamide
3-[(4aR,7aS)-4-(cyclohexylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
1-[(1R,5S,6R)-6-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}methyl)-3-azabicyclo[3.1.0]hexan-3-yl]butan-1-one
5-[1-(3,4-dimethoxyphenyl)propan-2-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
(1R,5R)-6-(cyclobutylmethyl)-3-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
2-cyclopropyl-8-[4-(1H-pyrazol-3-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1,3-oxazole-4-carboxamide
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-[(2-amino-1,3-thiazol-4-yl)methyl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
N-(2-hydroxy-2-phenylethyl)-N-methyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
(3S,4R)-4-phenyl-1-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetyl)pyrrolidine-3-carboxylic acid
7-[(3-methoxyphenyl)methyl]-2-[2-(methylsulfanyl)pyrimidin-4-yl]-2,7-diazaspiro[4.5]decane
4-benzyl-1-[4-(1H-pyrazol-1-yl)benzoyl]-1,4-diazepan-5-one
(3aR,5R,6S,7aS)-2-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-octahydro-1H-isoindole-5,6-diol
1-{3-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
ethyl 3-{[2-(4-chlorophenyl)morpholine-4-carbonyl]amino}propanoate
2-amino-4-(5-hydroxy-2-methoxyphenyl)-6-(4-hydroxyphenyl)-5-methylpyridine-3-carbonitrile
(1R,5R)-6-methyl-3-(2-phenoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonane
3-[(2R,3R,6R)-5-(2H-1,3-benzodioxol-5-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
(1R,5R)-6-benzyl-3-(2-butoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonane
1-(2-{[5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)piperidine-3-carboxamide
N-[(3R,4S)-1-[(dimethyl-4H-1,2,4-triazol-3-yl)methyl]-4-propylpyrrolidin-3-yl]cyclobutanecarboxamide
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl){[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}amine
6-[4-fluoro-3-(hydroxymethyl)phenyl]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
(2R)-1-({4-[(6-methoxypyridin-3-yl)carbamoyl]phenyl}methyl)pyrrolidine-2-carboxamide
4-{2-[(2S)-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]-2-oxoethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
2-(3-{[(1-hydroxybutan-2-yl)(thiophen-3-ylmethyl)amino]methyl}-1H-indol-1-yl)acetamide
1-({3-[2-(methoxymethyl)piperidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-indole
4-(cyclopropylmethyl)-1-(isoquinoline-1-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(2,3,6-trifluorophenyl)methyl]piperidin-3-yl}propanamide
4-[4-(4-chlorophenyl)butanoyl]-N,N-dimethylpiperazine-1-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)acetamide
(1S,6R)-3-methyl-9-[4-(1H-pyrazol-5-yl)benzoyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-{2-[3-(5-methylpyridin-2-yl)-1-(thiomorpholin-4-yl)prop-2-yn-1-yl]phenoxy}ethan-1-ol
2-{5-[2-(1H-imidazol-2-yl)benzoyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-1,2,3,4-tetrahydroisoquinoline
2-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)quinolin-8-ol
6-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-(2-{2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1H-imidazol-1-yl}ethyl)pyridine
1-[(2-methoxy-5-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}phenyl)methyl]-1H-pyrazole
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}furan-3-carboxamide
N-(3,3-diphenylpropyl)-6-(quinolin-5-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
2-[2-(adamantan-1-ylsulfanyl)acetamido]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetic acid