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2-[1-(2-propoxyphenyl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(4aS,8aS)-2-(5-chloro-3-fluoropyridin-2-yl)-decahydro-2,7-naphthyridin-4a-ol
N-[3-(cyclohexyloxy)propyl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
3-(2-methoxyphenyl)-4-(1-phenylethyl)-4H-1,2,4-triazole
6-methyl-4-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1,2-dihydropyridin-2-one
2-(2-{[(2-chlorophenyl)methyl]sulfanyl}acetyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(4aS,8aR)-1-(2-aminoethyl)-6-[2-(4-chloro-3-methyl-1H-pyrazol-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
1-[4-(2-methoxybenzoyl)piperazin-1-yl]-3-(pyridin-3-yl)propan-1-one
N-{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}-N-(prop-2-yn-1-yl)cyclohexanamine
1-methyl-4-(2-methyl-1,8-naphthyridine-3-carbonyl)piperazin-2-one
6-(5-chlorothiophene-2-carbonyl)-2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-(2-fluoro-4-methylbenzoyl)-3-(3-methoxyphenoxymethyl)piperidine
N-[(2-methyl-1H-indol-5-yl)methyl]-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
N-cyclooctyl-6-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-2-oxo-7-(pyrrolidin-1-yl)-1,2,3,4-tetrahydroquinoline-6-carboxamide
1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}azetidin-3-ol
{3-[4-chloro-2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1H-1,2,4-triazol-5-yl}methanol
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N,2-dimethylfuran-3-carboxamide
methyl 1-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-oxo-3-(pentan-3-yl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
5-ethyl-2-methyl-4-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-N-[(5-methylpyrazin-2-yl)methyl]acetamide
6-{3-[3-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-oxopropyl}-2,3,4,5-tetrahydropyridazin-3-one
2-[3-(1H-imidazol-1-yl)propyl]-9-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[1-(propan-2-yl)-1H-imidazol-2-yl]-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidine
5-benzyl-5-[1-({4-[methyl(phenyl)amino]phenyl}methyl)piperidin-4-yl]imidazolidine-2,4-dione
5-{1-[(6-chloro-2H-chromen-3-yl)methyl]pyrrolidin-2-yl}-3-methyl-1H-1,2,4-triazole
N-[2-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidin-1-yl)-2-oxoethyl]acetamide
3-{[3-(3-hydroxypiperidin-1-yl)propyl]carbamoyl}benzoic acid
5-[4-(aminomethyl)piperidin-1-yl]-2-({6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2,3-dihydropyridazin-3-one
7-methoxy-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{1-[(4-fluorophenyl)methyl]-7-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
1-(2-benzylmorpholin-4-yl)but-3-en-1-one
3-(2-methylpropyl)-N-[3-(methylsulfanyl)propyl]-1,2-oxazole-5-carboxamide
7-fluoro-3-({[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]amino}methyl)-1-(2-phenylethyl)-1,2-dihydroquinolin-2-one
(1R,5R)-N,N-dimethyl-6-(2-methyl-1H-pyrrole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-(morpholin-2-yl)-1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]ethan-1-one
2-[(2-ethoxyacetamido)methyl]-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
2-(2-fluorophenoxymethyl)-4-(1,2-oxazolidine-2-carbonyl)-1,3-oxazole
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-[2-(1H-pyrazol-1-yl)benzoyl]piperidine
2-amino-6-(4-hydroxyphenyl)-4-[2-(2-methoxyethyl)pyrimidin-5-yl]-5-methylpyridine-3-carbonitrile
2-(2-methoxyethyl)-8-{2-[methyl(phenyl)amino]acetyl}-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(2-methyl-1H-indol-1-yl)ethyl]-6-oxo-1-(2-phenylethyl)piperidine-3-carboxamide
1-cyclohexyl-3-(cyclopropylmethyl)-N-[2-(1H-imidazol-4-yl)ethyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}propane-1-sulfonamide
N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
2-(3-methyl-1H-1,2,4-triazol-5-yl)-N-[2-(5-methylfuran-2-yl)phenyl]pyrrolidine-1-carboxamide
1-(benzenesulfonyl)-N-(cyclohex-1-en-1-ylmethyl)cyclopropane-1-carboxamide
1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-3-[(3S,4R)-1-(propan-2-yl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propan-1-one
N-[2-(3-methoxyphenyl)phenyl]-1-(thiophen-2-ylmethyl)piperidine-4-carboxamide