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N-[(2,5-difluorophenyl)methyl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
1-(2-{[ethyl(2-hydroxyethyl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
1-[2-(azepan-1-yl)acetyl]-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
N-(5-chloro-2-methoxyphenyl)-3-{[(5-methyl-1,2-oxazol-3-yl)formamido]methyl}piperidine-1-carboxamide
(1R,3S)-7-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-3-ethoxy-7-azaspiro[3.5]nonan-1-ol
2-methyl-4-(1-{[5-(oxan-2-yl)thiophen-2-yl]methyl}piperidin-4-yl)pyrimidine
6-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-2-carboxylic acid
(2S,4S)-4-amino-N,N-diethyl-1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]pyrrolidine-2-carboxamide
3-(4-{[5-(2-methylpropyl)thiophen-2-yl]methyl}piperazin-1-yl)propan-1-ol
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
4-(5-methylpyridin-2-yl)-1-[2-(propan-2-yl)pyrimidine-4-carbonyl]piperidin-4-ol
1-(4-chlorophenyl)-3-cyclopropyl-5-{[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-1H-1,2,4-triazole
(oxolan-2-ylmethyl)(pyridin-4-ylmethyl){[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}amine
2-(2-chlorophenyl)-2-{[1-(propan-2-yl)piperidin-4-yl]formamido}acetic acid
1-(2-{1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(1-propyl-1H-pyrazol-4-yl)methyl]piperidin-2-one
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-[(1-phenylcyclohexyl)methyl]piperidine-3-carboxamide
4-methyl-3-oxo-N-(3-phenyl-1,2,4-thiadiazol-5-yl)-2-(propan-2-yl)piperazine-1-carboxamide
5-[(1S,5R)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]thiophene-2-carboxylic acid
1-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(pyrrolidin-1-yl)piperidine
N-(2-chlorophenyl)-4-(pyrrolidine-1-sulfonyl)piperazine-1-carboxamide
1-(5-acetylthiophene-3-carbonyl)-4-phenylpiperidine-4-carbonitrile
(2S,4R)-N-ethyl-4-[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[3-(pyridin-3-yl)propanoyl]pyrrolidin-3-yl]acetamide
N2-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)pyrimidine-2,4-diamine
2-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrazine
(3S,4R)-1-cyclopentyl-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
N-{1-[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
2-[(E)-2-cyclohexylethenyl]-6,7-dimethoxyquinazolin-4-amine
1-(2-aminoethyl)-4-benzyl-3-ethyl-1,4-diazepan-5-one
5-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole
2-{2-methoxy-5-[(4-phenyl-1,4-diazepan-1-yl)methyl]phenoxy}acetic acid
4-[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]-6-hydroxy-7-methoxy-1,2,3,4-tetrahydroquinolin-2-one
3-{4-[(2-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}propanamide
5-{methyl[(3-phenyl-1H-pyrazol-4-yl)methyl]carbamoyl}-2,1,3-benzoxadiazol-1-ium-1-olate
1-[1-(9H-purin-6-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
4-({2-[1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-(2-methoxyethyl)-1-methyl-N-(1-methylpiperidin-4-yl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-[5-(4-ethoxyphenyl)furan-2-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-(2,5-dihydro-1H-pyrrol-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine
N,1-dimethyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrrole-2-carboxamide
7-fluoro-2-methyl-N-[1-(pyrimidin-2-yl)piperidin-3-yl]quinoline-4-carboxamide
(5-{[methyl({2-[2-(prop-2-en-1-yl)phenoxy]ethyl})amino]methyl}furan-2-yl)methanol
(1S,5R)-3-[2-(2-fluorophenyl)acetyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
({5-[3-(2-methoxyphenyl)phenyl]-1,2,4-oxadiazol-3-yl}methyl)dimethylamine
2-[1-(1-benzofuran-3-carbonyl)piperidin-4-yl]-5-fluoro-1H-1,3-benzodiazole
3-({[(4-chlorophenyl)methyl]amino}methyl)-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
1'-(oxolan-3-ylmethyl)-1,2-dihydrospiro[indole-3,4'-piperidine]
3-{[2-(1-carboxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]methyl}benzoic acid