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N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(pyrazine-2-carbonyl)piperidin-3-amine
1-methyl-4-{[4-phenyl-5-(2-phenylethyl)-1H-imidazol-1-yl]methyl}pyrrolidin-2-one
(2S,4S)-4-amino-N-methyl-1-(naphthalene-1-carbonyl)pyrrolidine-2-carboxamide
5-{[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]sulfonyl}-2-methoxy-N-methylbenzamide
4-{[2-(1-cyclopropanecarbonylpiperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
1-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
(4aS,7aR)-1-(3-ethyl-1,2-oxazole-5-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-cyclobutyl-3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-(4-methanesulfonyl-1,4-diazepan-1-yl)propan-1-one
7-chloro-3,5-dimethyl-N-[3-(propan-2-yloxy)propyl]-1-benzofuran-2-carboxamide
N3-(butan-2-yl)-1-cyclopentyl-N5-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-(2-{3,9-diazaspiro[5.5]undecan-3-yl}-2-oxoethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
3-ethoxy-1-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
1-(2-{4-[1-(dimethylamino)ethyl]piperidin-1-yl}-2-oxoethyl)-3-methyl-1,2,3,4-tetrahydroquinazolin-2-one
2-{4-[1-(2-fluorophenyl)piperidin-4-yl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
N-{2-oxo-2-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethyl}benzamide
1-[2-(pyridin-4-yl)-4-{[(2R)-pyrrolidin-2-ylmethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
6-[4-(pyrimidin-5-ylmethyl)piperazin-1-yl]pyridine-3-carboxamide
2-amino-1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-2-methylpropan-1-one
N-[(2S,4R,6R)-2-(2-ethyl-4-methyl-1H-imidazol-5-yl)-6-(propan-2-yl)oxan-4-yl]benzamide
[1-(4-{4-[(adamantan-2-ylmethyl)amino]piperidin-1-yl}benzoyl)piperidin-3-yl]methanol
(2S,4S)-4-amino-N,N-diethyl-1-[2-(pyridin-4-ylsulfanyl)acetyl]pyrrolidine-2-carboxamide
4-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-1-(2-methoxyphenyl)-5-methylpiperazin-2-one
2-(benzyloxy)-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methylacetamide
2-[(4aR,7aS)-4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
N-methyl-N-{1-[1-(oxolane-2-carbonyl)piperidin-4-yl]-2-phenylethyl}pyridine-2-carboxamide
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3,3,3-trifluoropropanamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-(2-methyl-1,4-oxazepane-4-carbonyl)-N-(1,2-oxazol-3-ylmethyl)benzene-1-sulfonamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[3-(methylsulfanyl)butyl]piperazine
(1S,5R)-6-benzyl-3-(6-hydroxyhexyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(1H-indazol-6-yl)-4-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-2-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-3-propyl-1H-pyrazole-5-carboxamide
1-[(2-fluorophenyl)methyl]-N-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-amine
1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-({[(2-methylphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
[(8-chloroquinolin-2-yl)methyl](methyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(5-oxopyrrolidin-2-yl)acetamide
3-(4-methyl-1H-pyrazol-1-yl)-1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]propan-1-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-3-(1,2-oxazolidin-2-yl)propanamide
N-({5-methyl-2-[3-(2-methylfuran-3-amido)phenyl]-1,3-oxazol-4-yl}methyl)-3-phenyl-1H-pyrazole-5-carboxamide
4-{[2-(dimethylamino)-6-ethylpyrimidin-4-yl]amino}-1-[(3-fluorophenyl)methyl]pyrrolidin-2-one
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-(propan-2-yl)-4-{[3-(pyrrolidin-1-yl)propyl]sulfamoyl}benzamide
4-({4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-2-methoxyphenol
N-methyl-2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}acetamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-3-(2-oxopyrrolidin-1-yl)propanamide
3-fluoro-N-{[2-(trifluoromethyl)phenyl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
N,4-dimethyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-2-amine
2-methyl-6-(quinoxalin-2-yl)-3,4-dihydroquinazolin-4-one