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5-(1-ethyl-1H-imidazol-5-yl)-1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4-phenyl-1H-imidazole
6-methyl-2-({2-[4-(1-phenylethyl)-1H-1,2,3-triazol-1-yl]ethyl}amino)-3,4-dihydropyrimidin-4-one
6-(furan-2-yl)-2-[3-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
N-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
6-(2-fluoro-4-methoxyphenyl)-7-methyl-2-[(3R)-3-methylpiperazine-1-carbonyl]-7H,8H-imidazo[1,2-a]pyrazin-8-one
4-(4-{2-azabicyclo[2.2.1]heptane-2-carbonyl}piperidin-1-yl)-2-(2H-1,3-benzodioxol-5-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-{1-[(6-chloro-2H-chromen-3-yl)methyl]piperidin-3-yl}-4-(2-methylphenyl)piperazine
4-[(4-methyl-5-{[(2E)-3-phenylprop-2-en-1-yl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]piperidine
1-[3-(methylsulfanyl)propyl]-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-methylbutanamide
4-methyl-N-{2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidin-2-amine
3-butyl-1-methyl-4-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperazin-2-one
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-[(3R,4S)-1-(1H-imidazol-2-ylmethyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
4-{8-methyl-3-[(4-methylpiperazin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carbonyl}morpholine
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(pent-2-yn-1-yl)piperidine
1-butyl-4-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)piperazin-2-one
N-methyl-1-propyl-N-[2-(pyridin-2-yl)ethyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{1-[(2-fluorophenyl)methyl]-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
6-[1-methyl-10-oxo-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-4-yl]pyridine-2-carbonitrile
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-(2,4-dimethoxyphenyl)-3-[ethyl(pyridin-4-ylmethyl)amino]piperidine-1-carboxamide
3-[(pyrazin-2-yl)amino]adamantan-1-ol
9-methoxy-7-(4-methylphenyl)-4-[(5-methylthiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(4aS,7aR)-1-[(4-fluoro-3-methylphenyl)methyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[2-(1H-imidazol-1-yl)ethyl]({[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]methyl})methylamine
methyl N-{[(2S,4S)-4-fluoro-1-[2-(5-oxo-2-phenylcyclopent-1-en-1-yl)acetyl]pyrrolidin-2-yl]methyl}carbamate
2-[(2S)-2-amino-3-hydroxypropanoyl]-N-[2-(pyridin-2-yl)ethyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-(1-benzylpyrrolidin-3-yl)-5-ethylpyrimidin-2-amine
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)[2-(1,3-thiazol-4-yl)ethyl]amine
4-{2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl}-6-methyl-1,2-dihydropyridin-2-one
1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-4-(hydroxymethyl)azepan-4-ol
N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
5-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(2,5-dihydroxy-2-methylpentyl)-1-[4-(furan-2-yl)phenyl]urea
3-{1-[(2S,4R)-4-aminopyrrolidine-2-carbonyl]piperidin-4-yl}phenol
3-{1-[(4-chlorophenyl)methyl]-3-methyl-1H-pyrazol-5-yl}-1-(oxolan-2-ylmethyl)urea
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-(pyridin-4-yl)propan-1-one
(2S,4R)-1-benzyl-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
4-(3,6-dimethyl-1-benzofuran-2-carbonyl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
4-{2-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
7-{[(4-methyl-1,3-thiazol-2-yl)carbamoyl]carbonyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1,3-benzoxazol-2-yl)piperidin-3-ol
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-(2-methoxyethyl)-1-methylpiperidin-4-amine
2-(1H-pyrazol-1-ylmethyl)-4-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-1,4-oxazepane
1-{4-[(5-aminopentyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-{1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-methyl-1-oxobutan-2-yl}acetamide
9-[(3-fluoro-5-methylphenyl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine