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N-methyl-2-[2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamido]acetamide
3-[2-(4-benzylpiperidin-1-yl)-2-oxoethyl]-4-[(2,3-difluorophenyl)methyl]piperazin-2-one
N-[(3R,4S)-4-cyclopropyl-1-[1-(3-methylphenyl)piperidin-4-yl]pyrrolidin-3-yl]-2-hydroxyacetamide
9-[2-(4-hydroxyphenyl)acetyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
[(1,5-dimethyl-1H-indazol-3-yl)methyl][1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amine
2-hydroxy-1-(6-hydroxy-4-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
N-[(2R,3R)-2-methoxy-1'-[(5-methylfuran-2-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
6-(4-fluorophenyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-3-(piperidin-4-ylmethyl)benzamide
2-(cyclohexylmethyl)-4-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}morpholine
4-[1-(dimethylsulfamoyl)piperidin-3-yl]benzoic acid
2-(2-fluorophenyl)-N-[2-(5-methyl-1,3-oxazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]acetamide
2-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-4H-chromen-4-one
N-benzyl-1-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
4-[3-(2,5-difluorobenzoyl)piperidin-1-yl]-6-(propan-2-yloxy)pyrimidin-2-amine
5-{4-[(3-cyanopiperidin-1-yl)methyl]-2-methoxyphenoxymethyl}furan-2-carboxylic acid
3-{[1-(1H-indole-2-carbonyl)piperidin-4-yl]methyl}benzoic acid
(3S,4R)-4-(pyridin-4-yl)-1-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
4-(benzyloxy)-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}butan-1-one
2-methyl-8-(4-phenylbenzenesulfonyl)-2,8-diazaspiro[4.5]decan-3-one
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
ethyl 4-(10-{[1-(furan-2-yl)ethyl]carbamoyl}-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-3-yl)piperidine-1-carboxylate
(3S,4S)-4-(4-methylpiperazin-1-yl)-1-{[2-(trifluoromethoxy)phenyl]methyl}pyrrolidin-3-ol
(2S)-1-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carbonyl}pyrrolidine-2-carboxamide
2-(1-methyl-1H-pyrazol-4-yl)-5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridine
N-cyclopentyl-1-{1-[(2,3-dimethoxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
N-[(3R,4R)-1-[2-(3-chlorophenyl)acetyl]-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
5-chloro-N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-[3-(oxan-4-yl)-5-[(1R,2R)-2-phenylcyclopropyl]-1H-1,2,4-triazol-1-yl]pyridine
N-[2-(4-fluorophenyl)-1-{1-[2-(phenylsulfanyl)acetyl]piperidin-4-yl}ethyl]-N-methyl-3-(methylsulfanyl)propanamide
3,5-dimethyl-2-[3-(pyridine-2-carbonyl)piperidine-1-carbonyl]-1H-indole
4-(2-hydroxy-5-methoxybenzoyl)-1-(3-methoxyphenyl)piperazin-2-one
1-(3-methylbut-2-en-1-yl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)-3,3-diethylpyrrolidine-1-carboxamide
(4aR,8aS)-1-(cyclohexylmethyl)-6-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-decahydro-1,6-naphthyridin-2-one
5-{[4-phenyl-5-(2,4,6-trimethylphenyl)-1H-imidazol-1-yl]methyl}-1H-1,2,3,4-tetrazole
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-{[2-(trifluoromethoxy)phenyl]methyl}urea
4-(3-{1-[(4-methyl-1,3-thiazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine
2-[4-(1-benzothiophen-3-yl)-2-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy]-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-4-(1H-pyrazol-3-yl)benzamide
3-[7-(2-chlorobenzamido)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]pyridin-1-ium-1-olate
4-[1-(1-methanesulfonylpiperidin-4-yl)piperidine-3-carbonyl]morpholine
2-(2-{[(1-hydroxybutan-2-yl)(pyridin-2-ylmethyl)amino]methyl}phenoxy)acetamide
1-(2H-1,3-benzodioxol-5-yl)-3-cyclopropyl-5-[2-(trimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazole
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
2-[4-(ethoxycarbonyl)piperazin-1-yl]-2-(trimethyl-1H-pyrazol-4-yl)acetic acid
1-(2-hydroxyethyl)-4-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-1,4-diazepan-6-ol
2-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-2,8-diazaspiro[4.5]decane