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2-{1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
1-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-3-(3-methoxyphenoxy)propan-2-ol
1-ethyl-3,5-dimethyl-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
4-[(4-methylphenyl)methyl]-3-{2-oxo-2-[4-(pyrrolidin-1-yl)piperidin-1-yl]ethyl}piperazin-2-one
1-[(3,5-dimethylfuran-2-yl)methyl]-3-phenylpyrrolidin-3-ol
(4aS,7aR)-1-(dimethyl-1,3-oxazole-4-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1,5-dimethyl-4-{[8-(2-methylquinolin-4-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}-1H-pyrrole-2-carbonitrile
N-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-1-(2-methylpropyl)piperidin-4-amine
(4aS,8aR)-6-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
3-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-N-[(1r,4r)-4-hydroxycyclohexyl]benzene-1-sulfonamide
1-{4-[2-(pyridin-4-yl)ethyl]piperazin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl](methyl)[(3-methylquinoxalin-2-yl)methyl]amine
1-{6-methylthieno[2,3-d]pyrimidin-4-yl}-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]piperidin-4-amine
2-cyclopentyl-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
5-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-2-amine
(4aS,7aR)-1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(2-methoxyethyl)-1-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}piperidine-3-carboxylic acid
methyl 5-oxo-5-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}pentanoate
3-(pyrrolidin-1-ylmethyl)-1-(thiophen-3-ylmethyl)piperidin-3-ol
2-(4-acetylphenoxy)-1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}ethan-1-one
N-(2-methoxyethyl)-3-(4-methoxyphenyl)-N-(1-methylpiperidin-4-yl)-1H-pyrazole-5-carboxamide
N-(3,3-diphenylpropyl)-6-[2-(1,3-thiazol-4-yl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
1-[4-({2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}amino)piperidin-1-yl]-2-methylpropan-1-one
N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
N,5-dimethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
2-amino-6-(2-methoxyphenyl)-4-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
7-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
5-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-3-ethyl-1,2-oxazole
N-benzyl-N-[(1R,2R)-2-hydroxycyclohexyl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
N-[2-(4-hydroxypiperidin-1-yl)-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl]thiophene-2-carboxamide
N-[4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]benzamide
2-(4-fluorophenyl)-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidine
2-ethyl-7-[6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-2,7-diazaspiro[4.4]nonane
2-[2-(8-chloroquinolin-2-yl)-1H-imidazol-1-yl]acetamide
N3-tert-butyl-1-cyclohexyl-N5-[2-(4-methoxyphenyl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1-(furan-2-ylmethyl)-1H-imidazole
ethyl 1-methyl-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
N-methyl-3-[(2-methylprop-2-en-1-yl)oxy]-N-[(3-methylpyridin-2-yl)methyl]benzamide
1-benzyl-8-[(4-methoxyphenyl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1-benzofuran-2-carboxamide
N-cyclopentyl-2-({[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}amino)propanamide
(3aS,7aR)-2-[2-(4,6-dimethyl-1-benzofuran-3-yl)acetyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-[2-methoxy-4-({[2-(pyridin-3-yloxy)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
N-{2-[1-(2-phenylethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
2-(3-chlorophenyl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
3-methyl-1-(1-{2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}piperidin-3-yl)butan-1-one
N-[3-(cyclopentyloxy)propyl]-3-(piperidin-3-yl)benzamide
4-[4-(morpholine-4-carbonyl)piperazine-1-carbonyl]-1,2-dihydroquinolin-2-one
6-[(3S,4R)-3-carboxy-4-(pyridin-4-yl)pyrrolidin-1-yl]pyridine-3-carboxylic acid