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(3S,4R)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
2-{[3-(4-hydroxyphenyl)-1H-pyrazol-5-yl]formamido}-3-phenylpropanoic acid
(3aR,6aS)-2-(cyclopropylmethyl)-5-[2-(morpholin-4-yl)acetyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2R,3R,6R)-5-(morpholine-4-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(1'-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)-2-methoxyethan-1-one
3-(3-{1-[2-(ethylsulfanyl)ethyl]-1H-pyrazol-3-yl}phenyl)pyrazine-2-carbonitrile
2-amino-4-(5-cyano-1-ethyl-1H-pyrrol-3-yl)-6-(4-hydroxyphenyl)pyridine-3-carbonitrile
4-[1-(2,5-dimethylfuran-3-carbonyl)pyrrolidin-3-yl]-1-(2-methylpropyl)piperidine
3-{[(1S,5R)-6-(cyclopropylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-7-methoxy-1,2-dihydroquinolin-2-one
2-(3-phenylpropyl)-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
1-[(4-methyl-1H-imidazol-2-yl)methyl]-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
(2S,4R)-4-amino-N-(propan-2-yl)-1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}pyrrolidine-2-carboxamide
N-{3-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-3-oxopropyl}methanesulfonamide
3-[1-methyl-3-(pyrimidin-2-yl)-1H-1,2,4-triazol-5-yl]-1,2,5,6,7,8-hexahydroquinolin-2-one
2-cyclopropyl-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]pyrimidine-5-carboxamide
4-[5-(1H-pyrazol-3-yl)furan-2-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(1S,5R)-3-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-5-propyl-1,3,4-oxadiazol-2-amine
3-[4-(pyridin-2-ylmethyl)piperazine-1-carbonyl]piperidine-1-carboxamide
N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
4-methoxy-3-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]benzene-1-sulfonamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,2,5-trimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
(2S)-2-[(2-ethylpyrimidin-5-yl)formamido]-4-methylpentanamide
3-{3-[1-(2-methoxyethyl)-1H-pyrazol-3-yl]phenyl}pyridine
N-[3-(azepan-1-yl)-2-hydroxypropyl]-1,7-dimethyl-1H-indole-2-carboxamide
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
4-(1-methyl-1H-imidazol-2-yl)-1-(3-phenyl-1H-pyrazole-4-carbonyl)piperidine
(4aR,7aS)-1-(2-methoxyethyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-cyclopropyl-N-ethyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-N-(2-hydroxyethyl)-1H-pyrazole-4-carboxamide
3-{[(2,4-dihydroxypyrimidin-5-yl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
4-[(diethylamino)methyl]-5-ethyl-N-{[(3R,4R)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}furan-2-carboxamide
1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)piperidine-3-carboxamide
{5-[2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
N-[(6-methylpyridin-2-yl)methyl]-7-(oxan-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-methyl-3-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
5-[4-(1H-imidazol-1-ylmethyl)phenyl]-2,3-dihydro-1H-isoindole
N-methyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[(5-propyl-1H-pyrazol-3-yl)methyl]acetamide
1,3-dimethyl-N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
[5-({[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)-2-(propan-2-yloxy)phenyl]methanol
2-[5-cyclopropyl-4-(4-ethylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-(thiophen-2-yl)pyrimidine
N-[2-({4-methyl-6H,7H,8H-cyclopenta[g]quinolin-2-yl}amino)ethyl]methanesulfonamide
3-{1-[2-(dimethylamino)-2-(4-methylphenyl)acetyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
1-[(3S,4R)-4-ethoxyoxolan-3-yl]-2-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazole
N-[(5-methylfuran-2-yl)methyl]-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-benzofuran-5-carboxamide
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl){[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
2-{4-[1-(morpholin-4-yl)ethyl]phenyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-(1-cycloheptylpiperidin-3-yl)-2-(3,4,5-trimethoxyphenyl)acetamide
{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
N-(6-phenoxypyridin-3-yl)-1-propylpiperidine-2-carboxamide