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5-(methoxymethyl)-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
8-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-3-ol
1-{1-[2-(2-chloro-6-fluorophenyl)acetyl]piperidin-3-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
1-(oxan-4-yl)-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]piperidine-3-carboxamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-5-(trifluoromethyl)pyridin-2-amine
5-(2-methylpropyl)-1'-(2-propyl-1,3-thiazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(5-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
4-({2-[3-(dimethylamino)propoxy]phenyl}methyl)-1-phenylpiperazin-2-one
6-[(diethylamino)methyl]-N-(2-methoxy-6-methylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-2-{pyrazolo[1,5-a]pyridin-7-yl}pyridine
(2S,4R)-4-amino-N-ethyl-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]pyrrolidine-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}furan-3-carboxamide
6-(4-{[1-(prop-2-en-1-yl)-1H-1,3-benzodiazol-2-yl]methyl}piperazin-1-yl)pyrimidine-2,4-diamine
4-{2-[(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)amino]ethyl}benzene-1-sulfonamide
8-fluoro-3-[2-(morpholin-4-yl)ethyl]-3,4-dihydroquinazolin-4-one
1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}-4-ethylpiperazine
[(2S,6S)-4-[4-(piperidin-1-yl)benzoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
7-(2-ethylbutyl)-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
2-{1-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]pyrrolidin-3-yl}benzoic acid
N-[1-(3,5-difluorophenyl)ethyl]-6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(3-chloro-4-methoxyphenyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-5-oxopyrrolidine-3-carboxamide
4-propyl-5-[2-(thiophen-2-yl)azetidine-1-carbonyl]pyrimidine
[3-(furan-2-carbonyl)-9-[(3-methyl-1,2-oxazol-5-yl)methyl]-3,9-diazaspiro[5.5]undecan-1-yl]methanol
methyl (2S,4S)-4-(2,5-dimethoxybenzenesulfonamido)-1-methylpyrrolidine-2-carboxylate
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)-1H-1,2,3-benzotriazole-5-carboxamide
methyl 1-ethoxy-8-[2-(5-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
2-[(3-ethoxypropanamido)methyl]-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
(3S,5R)-N3-butyl-N5-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]piperidine-3,5-dicarboxamide
2-(4-phenylpiperazine-1-carbonyl)-3,4-dihydroquinazolin-4-one
N-({1-[(2-methoxyquinolin-3-yl)methyl]piperidin-3-yl}methyl)acetamide
2-{2-[1-(2-ethoxyethyl)-4-phenyl-1H-imidazol-5-yl]-1H-pyrrol-1-yl}pyrimidine
6-(methoxymethyl)-1-methyl-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(3-chloro-1,2-oxazol-5-yl)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
2-(dimethylamino)-N-[3-(dimethylamino)-2,2-dimethylpropyl]-2-(2-methylphenyl)acetamide
4-{[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile
1-cyclohexanecarbonyl-N-[(4-hydroxy-3,5-dimethylpyridin-2-yl)methyl]pyrrolidine-2-carboxamide
2-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-6-phenylpyridine-3-carboxylic acid
5-[(4-fluorophenyl)methyl]-5-[1-(quinolin-4-yl)piperidin-4-yl]imidazolidine-2,4-dione
4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-1,4-oxazepan-6-ol
N-{[2-(azepan-1-yl)-7-methoxyquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-(2-{3-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)-3-methoxy-1,2-dihydropyridin-2-one
6-(2-fluoro-4-methoxyphenyl)-7-methyl-2-(2-methylpyrrolidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
(5-{[(furan-2-ylmethyl)(3-methylbutan-2-yl)amino]methyl}-2-methoxyphenyl)methanol
3-butyl-4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-1-methylpiperazin-2-one
1-(cyclopropylmethyl)-N-ethyl-5-[3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
8-[2-(4-fluorophenoxy)ethyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
(3S,4R)-N,N-dimethyl-4-(propan-2-yl)-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidin-3-amine
5-[({5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}(methyl)amino)methyl]-N-methylpyrimidin-2-amine