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4-[1-(propan-2-yl)-1H-imidazol-2-yl]-N-[4-(propan-2-yl)phenyl]piperidine-1-carboxamide
5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-N-(oxan-4-yl)pyrimidin-2-amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(3-chlorophenyl)-5,8-dimethoxyquinolin-3-yl]methyl}-2-methylpropanamide
1-(pyrimidin-2-yl)-N-[(2,3,6-trifluorophenyl)methyl]piperidin-3-amine
2-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-3,5-difluoropyridine
4-(hydroxymethyl)-3-(3-phenoxypropyl)-1,3-oxazolidin-2-one
N-(prop-2-en-1-yl)-2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
3-[1-(6-methylpyridin-2-yl)propan-2-yl]-1-[4-(2-oxopyrrolidin-1-yl)phenyl]urea
N-cyclooctyl-4-oxo-4-[2-(trifluoromethyl)pyrrolidin-1-yl]butanamide
1-(3-chlorophenyl)-4-(dimethyl-1,3-thiazole-5-carbonyl)-5-methylpiperazin-2-one
N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]thiophene-2-carboxamide
4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-N-{[3-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrimidin-2-amine
[(4-{[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl](methyl)(2-phenylethyl)amine
N3-[2-(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]piperidine-1,3-dicarboxamide
5-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-6-methyl-2-(2-methylpyrimidin-4-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
N-[1-(hydroxymethyl)cyclopentyl]-1-[(4-methylphenyl)methyl]-5-oxopyrrolidine-3-carboxamide
2-ethyl-9-[2-(3-methoxyphenoxy)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
6,6-dimethyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-5-oxothiomorpholine-3-carboxamide
5-(2,4-difluorophenoxymethyl)-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
methyl (2S)-2-({5-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazol-3-yl}formamido)propanoate
8-(2-methoxypyridine-4-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(4-methoxy-2-methylphenyl)benzamide
2-ethoxy-5-[2-(4-fluorophenyl)pyrimidin-4-yl]benzoic acid
1-{3-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
N-[3-methoxy-5-(trifluoromethyl)phenyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-(4-chloro-2-methoxy-5-methylphenyl)-3-[4-(oxolan-2-yl)butyl]urea
6-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(3,5-difluorophenyl)-6-(morpholin-4-yl)pyrimidin-2-amine
1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-2-methyl-2-(morpholin-4-yl)propan-1-one
9-(1H-pyrazole-4-sulfonyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
[(1-cyclopentylpiperidin-3-yl)methyl][3-(methylsulfanyl)propyl][2-(piperidin-1-yl)ethyl]amine
4-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]morpholine-2-carboxylic acid
2-[5-(hydroxymethyl)furan-2-yl]-1H-1,3-benzodiazole-5-carbonitrile
ethyl 1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
3-{imidazo[1,2-a]pyridin-2-yl}-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}propanamide
N-{2-oxo-2-[2-(3-phenylpropyl)morpholin-4-yl]ethyl}acetamide
methyl 2-{4-[(3,3-dimethylcyclohexyl)amino]piperidin-1-yl}acetate
{[7-chloro-2-(morpholin-4-yl)quinolin-3-yl]methyl}[2-(2-methoxyphenyl)ethyl]amine
N-[(1-ethyl-1H-indazol-3-yl)methyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
3-{[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-4-(propan-2-yl)piperazin-2-one
5-fluoro-N,N-dimethyl-2-[3-(1H-pyrazol-3-yl)phenyl]pyrimidin-4-amine
N-[2-(3-methylpyridin-2-yl)ethyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-{[3-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-{2-[cyclopentyl(methyl)amino]ethyl}-N,3,4,7-tetramethyl-1H-indole-2-carboxamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
(3R,4R)-7-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-3-(pyrrolidin-1-yl)-3,4-dihydro-2H-1-benzopyran-4-ol
N5-(cyclohexylmethyl)-N3-methyl-4-oxo-N3-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide