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N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]-3-phenyl-1H-pyrazole-4-carboxamide
2-(2-chloro-4-fluorophenoxymethyl)-4-(2-propylpyrrolidine-1-carbonyl)-1,3-oxazole
4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(2-hydroxyethyl)-1-[1-(5-methoxyfuran-2-carbonyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
1-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propan-1-one
2-(ethanesulfonyl)-1-(2-phenylethyl)-5-(pyrrolidin-1-ylmethyl)-1H-imidazole
N-(4-{[1-benzyl-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenyl)acetamide
(3R,4S)-1-(azepane-1-sulfonyl)-4-phenylpyrrolidin-3-amine
(1R,3S)-7-(3-chloro-4-methoxybenzoyl)-7-azaspiro[3.5]nonane-1,3-diol
9-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(2-methoxyethyl)-N-(2-methoxyphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
3-(2-{3-[(2-fluorophenyl)methoxy]azetidin-1-yl}-2-oxoethyl)-3,4-dihydroquinazolin-4-one
5-methyl-4-[(1S,5S)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyrimidin-2-amine
N-[(2,3-dimethylphenyl)methyl]-N-methyl-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]acetamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-{1-[2-(furan-2-yl)ethyl]-1H-imidazol-2-yl}-N-methylbenzene-1-sulfonamide
6-(2-chlorophenyl)-2-[4-(morpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
1-{2-[3-(2-ethylphenoxy)azetidin-1-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
2-(4-hydroxy-4-phenylpiperidin-1-yl)-2-(4-methoxy-2-methylphenyl)acetic acid
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]imidazo[1,2-a]pyridine-3-carboxamide
2-(1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidin-2-yl)pyridine
1-propyl-4-{[5-(pyrrolidin-3-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidine
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-cycloheptyl-1-cyclopropyl-4-oxo-5-(3-phenylpiperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
4-(3-methyl-3-phenylpiperidine-1-carbonyl)pyridin-2-amine
5-{5-methyl-[1,2,4]triazolo[4,3-a]pyridin-3-yl}-2-(propan-2-yl)pyrimidine
5-methyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}pyrazine-2-carboxamide
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-3-(pyridin-4-yl)propanamide
(1R,3S)-7-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]-3-methoxy-7-azaspiro[3.5]nonan-1-ol
(1r,4r)-4-{[4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}cyclohexan-1-ol
3-{1-[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(3-fluorophenyl)urea
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-(1-methylcyclopropanecarbonyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
2-{4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]morpholin-3-yl}acetic acid
2-amino-4-{[2-(pyrrolidin-1-yl)ethyl]amino}quinazoline-6-carboxylic acid
4-hydroxy-2-{[(2,2,6,6-tetramethylpiperidin-4-yl)amino]methyl}quinoline-6-carboxamide
3-methyl-1-(4-methyl-2-oxo-1,2-dihydroquinolin-7-yl)-3-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}urea
(2S)-2-{2-[2-methyl-4-oxo-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamido}propanamide
4-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-1-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
(3S,4S)-4-cyclopropyl-1-(2-methyl-5-propylpyrimidin-4-yl)pyrrolidine-3-carboxylic acid
methyl (2S,4R)-1-methyl-4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-amido]pyrrolidine-2-carboxylate
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(furan-2-yl)-1H-pyrazole-4-carbonyl)-N,N-diethylpyrrolidin-3-amine
(4aS,8aR)-1-(3-aminopropyl)-6-(2,1,3-benzothiadiazol-5-ylmethyl)-decahydro-1,6-naphthyridin-2-one
2-(9-{[(furan-2-ylmethyl)carbamoyl]methyl}-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl)propanoic acid
2-(4-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-1-(3-methylbut-2-en-1-yl)piperazin-2-yl)ethan-1-ol
N-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-2-[methyl(piperidin-4-yl)amino]acetamide
N-[(2,6-difluoro-3-methylphenyl)methyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
5-(morpholin-4-ylmethyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]furan-3-carboxamide
N-cyclooctyl-2-({2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}amino)acetamide
4-(ethoxymethyl)-1-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]piperidine
N-(2,3-dimethylphenyl)-N'-[2-(4-methylmorpholin-2-yl)ethyl]propanediamide