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4-(5-fluoro-2-methylbenzoyl)-1-(4-methylphenyl)piperazin-2-one
3-chloro-N-(2-methoxyethyl)-4-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
[3-(hydroxymethyl)-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-3-yl]methanol
4-(2-methoxyphenoxy)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidine
3-[(3-methoxyphenyl)methyl]-5-(oxolan-3-yl)-1,2,4-oxadiazole
3-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]-2-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-4-one
1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-3-(4-methylphenoxymethyl)piperidine
5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine
7-(5-methylthiophen-2-yl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-(1-methyl-1H-indazol-5-yl)urea
7-[3-(4-chlorophenyl)propyl]-2-oxa-7-azaspiro[4.5]decan-8-one
3-(2-hydroxyphenyl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
3-methyl-5-{2-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-(pyridin-2-ylmethyl)piperidin-4-amine
5-oxo-N-(4-phenoxyphenyl)-1,4,9-triazaspiro[5.5]undecane-9-carboxamide
N-methyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}thiophene-3-carboxamide
methyl({[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl})(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
5-methyl-4-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-4-yl}pyrimidine
3-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-1-[4-(2-oxopyrrolidin-1-yl)phenyl]urea
6,7-dimethoxy-4-methyl-2-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]quinoline
2-(2-chlorophenoxy)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
(9aR)-8-[(2-fluoro-5-methylphenyl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(butan-2-yl)-3-hydroxy-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N,4-dimethyl-2-phenylpyrimidine-5-carboxamide
(2R,4R)-N-(1-benzothiophen-2-ylmethyl)-4-hydroxy-N-methylpyrrolidine-2-carboxamide
({[1-(1H-1,3-benzodiazol-2-ylmethyl)pyrrolidin-3-yl]methyl}sulfamoyl)dimethylamine
(1S,9aR)-1-{[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-octahydro-1H-quinolizine
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
4-(1,1-dioxo-1λ6-thiolane-3-amido)-N-phenylpiperidine-1-carboxamide
N-benzyl-6-[4-(pyridin-2-ylmethyl)piperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-[(1-methylpiperidin-3-yl)methyl]-1,2-dihydroquinoxalin-2-one
N-[4-(2-hydroxyethyl)phenyl]-3-{[methyl(prop-2-en-1-yl)amino]methyl}benzamide
N-[2-(methylsulfanyl)ethyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
2-[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]-N-(oxolan-2-ylmethyl)acetamide
4-(2-fluorophenyl)-N-[(1s,4s)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexyl]benzamide
1-(2-hydroxy-3-methylbutanoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-3-[(3-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-methyl-3-[methyl({[1-(propan-2-yl)-1H-imidazol-5-yl]methyl})amino]butanamide
N-[(3R,4S)-4-cyclopropyl-1-[5-fluoro-4-(methylamino)pyrimidin-2-yl]pyrrolidin-3-yl]-3-(methylsulfanyl)propanamide
N-[(1S,2R)-2-[(2,3-dihydro-1H-inden-2-yl)amino]cyclobutyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
2-[2-methyl-3-({[3-(pyrrolidin-1-yl)propyl]amino}methyl)-1H-indol-1-yl]acetamide
3-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]-4-fluorobenzene-1-sulfonamide
N,5,6-trimethyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2-(pyrrolidin-1-yl)pyrimidin-4-amine
4-(2-fluoro-5-methoxyphenyl)-2-oxo-7-(pyrrolidin-1-yl)-1,2,3,4-tetrahydroquinoline-6-carboxamide
N-(3-methoxy-2,2-dimethylpropyl)-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(5-chloro-6-hydroxy-2-methylpyrimidin-4-yl)benzamide
5-(methoxymethyl)-N-[2-(3-phenylpiperidin-1-yl)ethyl]thiophene-2-carboxamide
N-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-chloro-N-cyclopropyl-N-({4-methoxy-3-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)benzamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-(propan-2-yl)-1,2-oxazole-3-carboxamide