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5-(naphthalen-1-yl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]-1,2,4-triazin-3-amine
2-(cyclopentylmethyl)-N-[3-(dimethylamino)-2,2-dimethylpropyl]-1,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[4-(quinazolin-4-yl)piperazin-1-yl]propan-1-one
1-(2-hydroxyethyl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)piperidine-3-carboxamide
{1-[4-(hydroxymethyl)benzoyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-cyclopentyl-N3-ethyl-N5-[furan-2-yl(phenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-(1,4-dioxan-2-ylmethyl)-3-[(1H-imidazol-2-ylmethyl)sulfamoyl]benzamide
1-(3-ethylpiperazin-1-yl)-2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethan-1-one
methyl 9-(cyclopentyloxy)-7-oxo-3-[3-(pyridin-3-yl)propanoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
8-[(2R,3S)-2-amino-3-hydroxybutanoyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
4-methyl-2-[1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
2-methyl-N-{[3-methyl-7-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1,3-thiazole-4-carboxamide
2-(3-chloro-4-fluorophenyl)-2-{[1-(propan-2-yl)piperidin-4-yl]formamido}acetic acid
2-(cyclopentylmethyl)-N-(3-methoxypropyl)-6-methyl-4-oxo-1-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]-N-[2-(propan-2-yloxy)ethyl]propanamide
3-cyclopropyl-N-(furan-2-ylmethyl)-1H-pyrazole-5-carboxamide
3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}propanamide
N,N-diethyl-3-(5-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-3-(pyrrolidin-1-yl)piperidine
6-methoxy-1-methyl-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)-1H-indole-2-carboxamide
N-tert-butyl-2-methyl-3-{[methyl(oxan-2-ylmethyl)carbamoyl]amino}benzamide
3-{2-[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]-2-oxoethyl}-1,3-thiazolidine-2,4-dione
N-[(2-ethoxyphenyl)methyl]-N-ethyl-2-(1-methylpiperidin-2-yl)acetamide
2-methyl-4-(4-{[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenyl)butan-2-ol
1-(4-{[4-(2-hydroxypropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
N-[2-(1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)ethyl]acetamide
N,2-dimethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]thieno[2,3-d]pyrimidin-4-amine
8-fluoro-2-(thiomorpholine-4-carbonyl)quinoline
N-{3-[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]propyl}acetamide
4-(1-{1-[4-(3-fluorophenyl)phenyl]piperidin-4-yl}azetidin-3-yl)morpholine
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(azepan-1-yl)-3-[2-methoxy-4-({[2-(pyridin-3-yloxy)ethyl]amino}methyl)phenoxy]propan-2-ol
2-({[(3S,4S)-4-hydroxy-1-(propan-2-yl)pyrrolidin-3-yl]amino}methyl)-6-methylquinolin-4-ol
7-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidine
N1,N1-dimethyl-N4-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]piperidine-1,4-dicarboxamide
N-(oxolan-2-ylmethyl)-5-(propan-2-yl)-N-(pyridin-4-ylmethyl)-1,2-oxazole-3-carboxamide
methyl 2-{2-[1-(pyridin-3-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenoxy}acetate
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-methoxy-5-[({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}amino)methyl]phenol
1-ethyl-5-methyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-1H-pyrazole-4-carboxamide
2-(5-{[2-(3-fluorophenyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyrazine
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanamide
N-(dimethyl-1H-1,2,4-triazol-3-yl)-10-azabicyclo[4.3.1]decane-10-carboxamide
1-(2-aminoethyl)-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-1H-1,2,3-triazole-4-carboxamide
N-(2-methylphenyl)-3-oxo-3-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]propanamide
4-{[(prop-2-en-1-yl)(pyridin-3-ylmethyl)amino]methyl}benzonitrile
N1-(pyridin-3-yl)-N3-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}propane-1,3-diamine
N-[(3R,4S)-4-cyclopropyl-1-[3-(methylsulfanyl)propyl]pyrrolidin-3-yl]-1-methyl-1H-pyrazole-4-carboxamide