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{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}(methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
2-(2-methoxyphenyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
(1R,3S,5S)-8-(5-phenyl-1,2-oxazole-3-carbonyl)-8-azabicyclo[3.2.1]octan-3-ol
N-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-3-methylthiophene-2-carboxamide
(2R,4R)-4-hydroxy-N-{[3-(trifluoromethoxy)phenyl]methyl}pyrrolidine-2-carboxamide
N,2-dimethyl-2-(morpholin-4-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
N-[(2-methylphenyl)methyl]-2-(4-methylpiperazin-1-yl)-N-(prop-2-en-1-yl)propanamide
ethyl 2-({3-[4-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}amino)acetate
(3S,4R)-1-(6-fluoro-4-hydroxyquinoline-3-carbonyl)-4-methylpiperidine-3,4-diol
3-(4-fluorophenyl)-3-[2-(2-phenyl-1H-imidazol-1-yl)acetamido]propanoic acid
N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]cyclopent-1-ene-1-carboxamide
4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-(oxolane-2-carbonyl)piperidine
(4-methoxy-4-methylpentan-2-yl)[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
2-({1-[(3-chloro-4-hydroxyphenyl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-4-(thian-4-yl)piperazine
(3S,4S)-4-cyclopropyl-1-[(2-fluoro-5-methoxyphenyl)methyl]pyrrolidine-3-carboxylic acid
(2R,6R)-4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-3-(1H-imidazol-1-ylmethyl)piperidine
(3aS,7aR)-2-[2-(3-methoxyphenyl)acetyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-(4-{2-[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]-2-oxoethoxy}phenyl)propan-1-one
4-[(2-cyclopentyl-2-phenylethyl)amino]-1λ4-thian-1-one
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-3-(2-methyl-1H-imidazol-1-yl)butanamide
2-methyl-5-(2-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)-3,4-dihydropyrimidin-4-one
3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)-N-[2-(thiophen-2-yl)ethyl]propanamide
N,N-dimethyl-4-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]benzamide
2-(2-chloro-6-fluorophenyl)-1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]ethan-1-one
N,N,2-trimethyl-7-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-1,4-diazepane
2-cyclohexyl-1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]propan-1-one
1-methyl-4-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]piperazine-2-carboxylic acid
4-{[3-fluoro-2-(trifluoromethyl)phenyl]methyl}-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
methyl 2-(3-{[(1-benzylpiperidin-4-yl)amino]methyl}-7-chloro-2-oxo-1,2-dihydroquinolin-1-yl)acetate
N,N-diethyl-1-[4-(piperidin-1-ylmethyl)benzoyl]pyrrolidin-3-amine
4-[3-(3-methylbutyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]-4-oxobutanamide
1-[(1R,5S)-6-azabicyclo[3.2.1]octan-6-yl]-3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)propan-1-one
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(2,6-dimethylpyrimidine-4-carbonyl)piperidine-4-carboxamide
(1R,3S,5S)-8-{[3-chloro-5-ethoxy-4-(prop-2-en-1-yloxy)phenyl]methyl}-8-azabicyclo[3.2.1]octan-3-ol
4-[5-(cyclohexylsulfanyl)furan-2-yl]-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
methyl 3-[(thiophen-2-ylformamido)methyl]-5-[3-(trifluoromethyl)benzenesulfonamido]benzoate
8-[2-(2-chlorophenyl)acetyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]oxane-4-carbonitrile
1-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-5-(2-methylpropyl)-4-phenyl-1H-imidazole
3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
9-(cyclopropylmethyl)-4-[(dimethyl-1,3-thiazol-5-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-(1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}azetidin-3-yl)morpholine
N-(3-benzylphenyl)-3-(morpholin-4-yl)azetidine-1-carboxamide
3-(2-methyl-1,3-benzothiazol-6-yl)-1-{1-oxaspiro[4.4]nonan-3-yl}urea
1-{1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidin-3-yl}pyrrolidin-2-one
5-methyl-2-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidin-4-amine