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N-(1-methyl-1H-1,2,3-triazol-4-yl)-5-[1-(1-methyl-1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
2-methyl-4-{[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-imidazole
3-(dimethyl-1,2-oxazol-4-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]propan-1-one
1-{2-[1-(2-methyl-2,3-dihydro-1-benzofuran-5-carbonyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
5-[1-(2-methylpyridine-3-carbonyl)pyrrolidin-2-yl]-N-(1,3-thiazol-2-yl)thiophene-2-carboxamide
2-methyl-N-({3-methyl-7-[4-(2-methylpropyl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-3-carboxamide
4-{4-[(3-chloropyridin-4-yl)methyl]piperazin-1-yl}-2-methylquinoline
N-{1-[(3-methylphenyl)methyl]cyclopropyl}-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
4-{[2-(3-methoxypropyl)piperidin-1-yl]methyl}pyridine
6-methoxy-3-{[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydro-1H-indol-2-one
4-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)pyridin-1-ium-1-olate
2-(2-methyl-1,3-benzoxazole-6-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
ethyl 2-(4-methanesulfonamidopiperidin-1-yl)-1,3-oxazole-4-carboxylate
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-(3-methoxypropyl)pyrimidin-2-amine
2-(furan-2-yl)-5-({2-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)pyrimidine
4-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-3-yl)benzoic acid
N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyethyl)pyrrolidin-3-yl]benzenesulfonamide
5-(1H-indol-3-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{2-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
N-[(4-ethoxyphenyl)methyl]-2-methoxy-N-(2-methoxyethyl)-4-methyl-1,3-thiazole-5-carboxamide
3-[(3S,4R)-3-cyclopropyl-4-{[5-(propan-2-yl)pyrimidin-4-yl]amino}pyrrolidin-1-yl]propan-1-ol
1-[3-(piperidin-4-ylmethyl)benzoyl]-2-(pyrrolidin-1-ylmethyl)piperidine
2-[2-(4-ethylpiperazin-1-yl)-4-(morpholin-4-yl)pyrimidin-5-yl]-2-methylpropanoic acid
9-methoxy-7-(5-methylthiophen-2-yl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(4aS,7aR)-1-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{2-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propyl}pyridine
1'-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
2-[4-(1-methyl-1H-imidazol-2-yl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
3-(1-butyl-1H-imidazol-2-yl)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidine
1-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-3-yl}-4-(2-methoxyphenyl)piperazine
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)propanamide
N-cyclopropyl-1-{1-[(4-methyl-1,3-thiazol-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
3-({[(2,5-dimethylphenyl)methyl]amino}methyl)-3-hydroxy-1-[(3-methoxyphenyl)methyl]piperidin-2-one
(2S,4R)-1-[(2-chlorophenyl)methyl]-4-{[(2,5-difluorophenyl)methyl]amino}-N-ethylpyrrolidine-2-carboxamide
6-{1-oxa-8-azaspiro[4.5]decan-8-yl}pyridine-2-carbonitrile
6-methyl-N4-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}pyrimidine-2,4-diamine
3-{4-[(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}-1-methyl-1,2-dihydropyridin-2-one
1-[(4-fluorophenyl)methyl]-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}piperazin-2-one
3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]propan-1-one
propan-2-yl (1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
(2R)-N-[2-fluoro-5-(4H-1,2,4-triazol-4-yl)phenyl]-2-(hydroxymethyl)pyrrolidine-1-carboxamide
2-{4-[4-(1H-pyrrol-1-ylmethyl)benzoyl]morpholin-3-yl}acetic acid
N-[(1R,3S)-3-(phenylcarbamoyl)cyclopentyl]-3,4-dihydro-2H-1-benzopyran-6-carboxamide
6-(cyclooctylamino)-2-methylheptan-2-ol
N-[2-(2-methoxyphenyl)ethyl]-2-[2-(trifluoromethyl)pyrrolidin-1-yl]acetamide
(1S,5R)-3-cyclobutanecarbonyl-6-(pyridine-3-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
N-{1-[1-(1-methylcyclopropanecarbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
2-[4-({methyl[(1-methylpiperidin-2-yl)methyl]amino}methyl)phenoxy]acetic acid