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2-(4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperazin-1-yl)-1-(pyrrolidin-1-yl)ethan-1-one
N3-cycloheptyl-1-cyclopropyl-N5-[2-(4-methoxyphenyl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-({cyclopropyl[(4-ethoxyphenyl)methyl]amino}methyl)-3-methoxyphenol
1-cyclohexyl-N3-[2-(1H-indol-3-yl)ethyl]-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-methyl-2-(piperidin-1-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}pyrimidine-5-carboxamide
5-[5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1H-indole
ethyl 1-[1-(pyridin-3-yl)propan-2-yl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-4-(pyrrolidin-1-yl)butan-1-one
2-(2-methoxyethyl)-8-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
N-butyl-N-methyl-2-[1-(3-methylphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
4-{[2-(4-methoxyphenyl)-1H-imidazol-1-yl]methyl}pyrimidine
3-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}pyrrolidin-3-ol
3-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl}-2,3-dihydro-1H-inden-1-one
(2R)-2-amino-1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(1H-indol-3-yl)propan-1-one
N-(2-chlorophenyl)-2-oxo-2-{2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}acetamide
3-(5-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
1-(carbamoylmethyl)-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]piperidine-3-carboxamide
2-(5-{[4-(1-methylpiperidin-4-yl)piperazin-1-yl]methyl}furan-2-yl)benzonitrile
(4aR,7aS)-4-(3-hydroxypyridine-2-carbonyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-{3-[5-(1-ethyl-1H-1,2,4-triazol-5-yl)-4-phenyl-1H-imidazol-1-yl]propyl}pyrrolidin-2-one
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-{3-[2-(1,4-oxazepan-4-yl)-2-oxoethyl]morpholin-4-yl}-4-(1H-pyrazol-4-yl)butan-1-one
3-methoxy-6-{3-[1-(3-methoxypropyl)-1H-pyrazol-3-yl]phenyl}pyridazine
6-(3-oxo-3-{3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidin-1-yl}propyl)-2,3,4,5-tetrahydropyridazin-3-one
9-(5-chloropyridine-2-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
3-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-1H-indole
1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(4-methanesulfonylphenyl)methyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
N-({5-[(2-methoxy-4-methylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
1-methyl-N-[1-(4-phenylphenyl)ethyl]piperidin-4-amine
N-[1-(4-chlorophenyl)cyclobutyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
2-(5-{2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazol-3-yl)pyridine
6-amino-N-[(1-benzylpiperidin-4-yl)methyl]-N-methylpyridine-3-carboxamide
8-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
4-[(1S)-1-cyclohexylethyl]-3-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2-(dimethylamino)-2-(3-fluorophenyl)acetamide
(3S,4S)-4-(4-fluorophenyl)-1-[1-(pyridine-3-carbonyl)piperidin-4-yl]piperidin-3-ol
2-{[1-(3-hydroxyadamantan-1-yl)ethyl]amino}propane-1,3-diol
1-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-2-(thiophen-2-yl)azetidine
1-(4-fluorobenzoyl)-4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
5-(1H-imidazol-1-ylmethyl)-2-[3-(2-methylphenoxy)azetidin-1-yl]pyridine
methyl[1-(4-methylpyridin-2-yl)propan-2-yl][(3-phenyl-1,2-oxazol-5-yl)methyl]amine
6-[4-(3-hydroxy-3-methylbutyl)benzoyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-(4-oxo-1,4-dihydropyridin-1-yl)acetamide
6-(piperidin-4-yl)-2-[2-(pyridin-2-yl)ethyl]-3,4-dihydropyrimidin-4-one
(3R,4R)-1-[(3-chloro-4-hydroxyphenyl)methyl]-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
(1R,2R,6S,7S)-4-[3-(1H-1,2,4-triazol-1-yl)adamantane-1-carbonyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane