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1-[(3-fluorophenyl)methyl]-4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine
(3S,4S)-1-[(3-chlorophenyl)methyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
1-[2-(2,4-dichlorophenoxy)acetyl]-N-ethylpyrrolidine-3-carboxamide
4-(1H-1,3-benzodiazol-2-ylmethyl)-1λ6-thiomorpholine-1,1-dione
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2,5-dimethyl-1,3-oxazole-4-carboxamide
8-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-(2,6-dimethoxy-4-methylphenyl)-2-[4-(pyrrolidin-1-yl)piperidin-1-yl]acetic acid
4-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-4-oxo-N-phenylbutanamide
2-(5-acetylthiophen-3-yl)-N-{1-[(4-methyl-1H-imidazol-5-yl)methyl]azepan-3-yl}acetamide
(4aS,8aR)-6-[(2-methyl-1,3-oxazol-4-yl)methyl]-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
4-(1-methyl-1H-imidazol-2-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
[(2S,6S)-4-[6-(trifluoromethyl)pyridin-2-yl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-(propan-2-ylsulfanyl)ethan-1-one
N,2-dimethyl-N-(quinolin-5-ylmethyl)-2-(thiophen-2-ylformamido)propanamide
N-[1-(pyridin-4-yl)propan-2-yl]-2-(2,3,6-trimethylphenoxy)acetamide
methyl (2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-(1-hydroxynaphthalene-2-amido)pyrrolidine-2-carboxylate
5-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N2-(2-methoxyethyl)-N4-[2-(1H-1,2,4-triazol-1-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-benzyl-4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
3-cyano-5-fluoro-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}benzamide
4-[9-(3-methylbutyl)-3,9-diazaspiro[5.5]undecane-3-carbonyl]benzonitrile
5-ethyl-N4,6-dimethyl-N4-[2-(oxan-4-yl)ethyl]pyrimidine-2,4-diamine
2-(3-methyl-1,2-oxazol-5-yl)-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethan-1-one
(2S,4R)-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}(2-methylpropyl)(pyridin-2-ylmethyl)amine
9-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
1-[3-(furan-2-yl)phenyl]-N-[2-(1H-pyrazol-1-yl)ethyl]piperidin-4-amine
2-propyl-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}pyridine-4-carboxamide
1-[(5-{1-[(2R)-2-hydroxy-2-phenylethyl]-1H-pyrazol-3-yl}thiophen-2-yl)methyl]piperidin-3-ol
1-ethyl-3-{2-oxo-2-[4-(pyrazin-2-yl)piperazin-1-yl]ethyl}-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
2-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-4H-chromen-4-one
1-({1-cyclohexyl-3-[hydroxy(phenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)pyrrolidin-2-one
N,N-dimethyl-3-[2-(1H-pyrrol-1-yl)benzamido]azepane-1-carboxamide
N-[2-(furan-2-yl)ethyl]-6-(morpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
6-[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-{3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-(5-hydroxy-4,4-dimethylpentyl)acetamide
1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-4-(1H-pyrrole-2-carbonyl)-1,4-diazepan-6-ol
2-phenyl-6-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}imidazo[1,2-a]pyridine
6-fluoro-2-({[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]amino}methyl)quinolin-4-ol
(1r,4r)-4-({methyl[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amino}methyl)cyclohexan-1-ol
2-(3,5-dimethyl-1H-pyrazol-4-yl)-7-(3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
8-(1H-indol-2-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3R,4R)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-(morpholin-4-yl)piperidin-3-ol
1-(1-cycloheptanecarbonylpiperidin-3-yl)-4-[3-(trifluoromethyl)phenyl]piperazine
1-ethyl-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}-5-oxopyrrolidine-3-carboxamide
3-[(2-amino-6-ethyl-5-methylpyrimidin-4-yl)amino]-1-(pyrrolidin-1-yl)propan-1-one
4-chloro-2-{[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]methyl}phenol
2-phenyl-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}imidazo[1,2-a]pyridine-6-carboxamide