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2-[(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-diethylacetamide
3-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
1-(1-{1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}ethyl)-4-methylpiperazine
methyl 1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidine-1-carbonyl]cyclopropane-1-carboxylate
2-(4-phenylpiperidin-1-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(3-methyl-1-benzothiophene-2-carbonyl)pyrrolidin-3-yl]methanol
1-ethyl-N-(3-hydroxypropyl)-2-oxo-N-(pyridin-4-ylmethyl)-1,2-dihydropyridine-4-carboxamide
(benzylsulfamoyl)[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]amine
3-(cyclopropylmethyl)-1-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxylic acid
(4aR,8aS)-1-(2H-1,3-benzodioxol-5-ylmethyl)-6-[2-(2,5-dimethoxyphenyl)acetyl]-decahydro-1,6-naphthyridin-2-one
3-{2-[4-(5,6-dimethylpyrimidin-4-yl)piperazin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
1-{1-[(2,5-dimethoxyphenyl)methyl]piperidin-3-yl}-4-(2-fluorophenyl)piperazine
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)-1-[(1R,4S)-7,7-dimethyl-2-oxobicyclo[2.2.1]heptan-1-yl]methanesulfonamide
(2S,4R)-4-{5H,6H-imidazo[2,1-b][1,3]thiazole-3-amido}-N-(propan-2-yl)-1-propylpyrrolidine-2-carboxamide
4-[8-(3-methoxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-2-carboxylic acid
3-[(3R,4S)-1-(dimethyl-1,3-oxazole-5-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1-ethylpiperidin-3-amine
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-3-hydroxy-2-methylbenzamide
(2S,4S)-N-ethyl-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-[(4,5-dimethylfuran-2-yl)methyl]-N-methylpiperidin-3-amine
1-{1,3-dioxo-2-[2-(1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}-N-[(1-hydroxycyclohexyl)methyl]piperidine-4-carboxamide
1-[(3,4-dimethylphenyl)amino]-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]cyclohexane-1-carboxamide
2-amino-5-methyl-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
6-ethoxy-2-{1-[(5-methyl-1,2-oxazol-3-yl)methyl]-1H-imidazol-2-yl}quinoline
1-(furan-2-ylmethyl)-4-[1-(methoxymethyl)cyclopropanecarbonyl]-1,4-diazepan-6-ol
1-[(3-methylfuran-2-yl)methyl]-4-phenylpiperidin-4-ol
2-(3-ethoxypropanoyl)-N-[(1-methylpiperidin-3-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
[(4S)-4-amino-5-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-5-oxopentyl]urea
3-[2-(1-cyclopentylpiperidin-2-yl)ethyl]-3H,4H-pyrido[4,3-d]pyrimidin-4-one
5-{1-[(2-hydroxy-6-methoxyphenyl)methyl]piperidin-4-yl}-5-propylimidazolidine-2,4-dione
N-{[(3S,4S)-3-hydroxy-1-[2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetyl]piperidin-4-yl]methyl}-3-methylbutanamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
ethyl 5-(1,3-benzothiazol-2-ylmethyl)-1-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-cyclobutaneamido-N-ethyl-N-(2-methylprop-2-en-1-yl)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
3-[4-phenyl-5-(2-phenyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]propan-1-ol
3-{[2-(pyrrolidin-1-yl)ethyl]sulfamoyl}-N-(2,2,2-trifluoroethyl)benzamide
(3S,4R)-1-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-({5-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
2-[methyl({[2-(thiophen-2-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl})amino]ethan-1-ol
N-[(3R,4R)-1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(methylsulfanyl)acetamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(furan-2-ylmethyl)-N-methylpiperidine-3-carboxamide
1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
4-(1H-indol-4-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[5-(3-fluoro-4-methoxyphenyl)-1H-indazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-(5-phenylpyridin-2-yl)acetamide
6-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
3-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-[3-(furan-2-yl)phenyl]urea
1-(2-methyl-1-benzofuran-5-carbonyl)-3-(propoxymethyl)pyrrolidine
1-({3-[3-(azocan-1-yl)-2-hydroxypropoxy]-4-methoxyphenyl}methyl)azetidin-3-ol