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3-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenol
2-(cyclopropylmethyl)-N-[3-(pyridin-3-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(2-chlorophenyl)methyl]-3-[1-(5-ethyl-1,2,4-oxadiazol-3-yl)piperidin-3-yl]propanamide
3-ethyl-3-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-4-yl}urea
N-(carbamoylmethyl)-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[(3R,4S)-4-cyclopropyl-1-(oxan-4-yl)pyrrolidin-3-yl]-3-(1H-1,2,4-triazol-1-yl)propanamide
2-({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)amino)ethan-1-ol
5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-2,3-dimethylbenzene-1-sulfonamide
7-fluoro-N-methyl-N-[(6-methylpyridin-2-yl)methyl]-2-(pyrimidin-5-yl)quinoline-4-carboxamide
4-{5-[(4-propylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-3-yl}benzoic acid
2-(4-fluoro-2-methoxyphenyl)-2-[4-(pyridin-3-yloxy)piperidin-1-yl]acetic acid
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-(2-oxopyrrolidin-1-yl)acetamide
3-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]benzonitrile
(4S)-4-phenyl-3-(pyridin-4-ylmethyl)-1,3-oxazolidin-2-one
N-[1-(azepan-1-yl)-2-methylpropan-2-yl]-3-(1H-imidazol-2-yl)benzamide
4-(1-methyl-1H-imidazol-2-yl)-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1H-1,2,3-triazole
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N,N-bis(2-hydroxyethyl)acetamide
1-{2-[methyl({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl})amino]ethyl}piperidin-2-one
1-[5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(methoxymethyl)piperidine
3-cyclopentaneamido-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
3,3,3-trifluoro-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
4-(2-methyl-1-phenyl-1H-1,3-benzodiazole-5-carbonyl)piperazine-2-carboxylic acid
5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-[(2,6-difluoro-3-methylphenyl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(1-methylpiperidin-4-yl)-2-(2-oxoazepan-1-yl)-N-(pyridin-4-ylmethyl)acetamide
(3S,7S)-5-[3-(1-methyl-1H-pyrazol-5-yl)propanoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-({5-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
2-[1-({3-methyl-1-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazol-4-yl}methyl)pyrrolidin-2-yl]pyridine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]propan-1-one
(4-{[(4,6-dimethoxypyrimidin-2-yl)(methyl)amino]methyl}oxan-4-yl)methanol
(4aS,8aR)-1-(2-phenylethyl)-6-(pyridin-4-yl)-decahydro-1,6-naphthyridin-2-one
3-[(2-fluorophenyl)formamido]-N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]propanamide
3-[6-amino-5-cyano-4-(4-methanesulfonylphenyl)pyridin-2-yl]benzoic acid
N-{4-[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]phenyl}acetamide
1-ethyl-4-[3-(2-phenylacetyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]acetamide
N-methyl-N-(pyrazin-2-ylmethyl)-2-[3-(trifluoromethyl)phenyl]acetamide
7-[(3,4-difluorophenyl)methyl]-2-(pyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N4-[2-(1H-indol-3-yl)ethyl]-N2,N2-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
3-(4-methoxyphenyl)-5-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]-1,2,4-oxadiazole
(1S,5R)-6-{pyrazolo[1,5-a]pyridine-3-carbonyl}-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
6-(benzyloxy)-4-[(3-hydroxy-4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,4-diazepan-2-one
2-amino-4-(2-methoxypyrimidin-5-yl)-5H,6H-furo[2,3-h]quinoline-3-carbonitrile
5-{4-[(6-chloropyridin-3-yl)methyl]piperazine-1-carbonyl}-N-ethylpyrimidin-2-amine
1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-2-(2,3,4-trifluorophenyl)ethan-1-one
3-benzyl-4-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazin-2-one
1-[2-fluoro-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}urea
methyl 3-benzamido-6-({methyl[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
3-[(1-acetylpiperidin-4-yl)oxy]-N-[(2-fluorophenyl)methyl]-4-methoxybenzamide
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-cycloheptanecarbonylpiperidine
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1-phenyl-1H-1,2,3-triazole-4-carboxamide