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4-fluoro-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
(1S,9S)-11-{2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
methyl 6-(2,4-difluorobenzoyl)-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(2S,4S)-4-amino-N-methyl-1-[4-(1,3-oxazol-5-yl)benzenesulfonyl]pyrrolidine-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-{2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
methyl 3-(4-acetyl-4-phenylpiperidine-1-carbonyl)benzoate
N-[2-(1H-1,3-benzodiazole-1-carbonyl)phenyl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
4-(2H-1,3-benzodioxol-5-yl)-3-cyclobutyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-({2-[(dimethylamino)methyl]phenyl}methyl)-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
2-methyl-1-{2-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1H-indole-3-carbonitrile
3-[1-butyl-5-(pyrrolidin-1-ylmethyl)-1H-1,2,4-triazol-3-yl]pyridine
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
2-cyclopropyl-1-[(4-fluorophenyl)methyl]-N,6-dimethyl-4-oxo-N-(thiophen-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-(2-methoxybenzoyl)-4-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperazine
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
5-[7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
3-hydroxy-1-(2-phenylethyl)-3-{[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]methyl}piperidin-2-one
methyl[(3-methyl-1H-pyrazol-5-yl)methyl]{[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
4-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
N-methyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-(oxan-2-ylmethyl)acetamide
1-benzyl-3-methyl-3-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)urea
(3S,4S)-1-[2-(3-methoxyphenyl)acetyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylquinoxaline-2-carboxamide
2-[(3,5-difluorophenyl)methyl]-8-[(2S)-3-hydroxy-2-methylpropyl]-2,8-diazaspiro[4.5]decan-3-one
2-({[5-(1-cyclohexanecarbonylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)ethan-1-ol
3-(2H-1,3-benzodioxol-5-yl)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}propanamide
2-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(4-methylpiperazin-1-yl)ethyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
6-{4-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-9H-purine
3-{[1-(piperidin-1-ylmethyl)cyclopropyl]sulfamoyl}-N-(prop-2-en-1-yl)benzamide
2-amino-6-{4-[(dimethylamino)methyl]thiophen-2-yl}-4-(3-ethyl-1H-pyrazol-5-yl)pyridine-3-carbonitrile
N-[3-(1H-imidazol-1-yl)propyl]-5-methyl-2-(propylamino)benzamide
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-{[(1,3-dimethyl-1H-pyrazol-5-yl)formamido]methyl}benzoate
2,2-dimethylpropyl 4-[(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-1-carboxylate
6-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-N,5-dimethylthieno[2,3-d]pyrimidin-4-amine
N-{3-[(1-methylpiperidin-4-yl)oxy]propyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-[3-(pyridin-4-yl)propyl]acetamide
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-4-(methylsulfanyl)benzamide
2-(2-methoxyquinolin-3-yl)pyridine-3-carbonitrile
dimethyl[(4-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-2-yl}phenyl)methyl]amine
ethyl (4aS,8aR)-6-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-decahydro-1,6-naphthyridine-4a-carboxylate
N-{2-[5-methyl-4-({methyl[1-(pyridin-3-yl)propan-2-yl]amino}methyl)-1,3-oxazol-2-yl]phenyl}methanesulfonamide
1-tert-butyl-3-(ethoxymethyl)-5-[(3-methoxyphenyl)methyl]-1H-1,2,4-triazole
N-(1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}azepan-3-yl)cyclopropanesulfonamide
4-(3-fluorobenzoyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-({1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}oxy)pyrimidine
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]pyrimidin-2-amine
(4aR,7aS)-1-[(5-methylfuran-2-yl)methyl]-4-(1H-pyrrole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione