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N-{[6-(1-benzothiophen-3-yl)pyridin-3-yl]methyl}acetamide
5-{2-[2-(3-methylbut-2-en-1-yl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-(1H-imidazol-2-ylmethyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-3-(2,5-dioxoimidazolidin-4-yl)propanamide
1-(4-{[ethyl(oxan-4-ylmethyl)amino]methyl}thiophen-2-yl)ethan-1-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1,3-oxazole-5-carboxamide
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-{2-[3-(methylsulfanyl)phenyl]acetyl}-decahydro-1,6-naphthyridin-2-one
1-(2-{1-[2-(3-chloro-4-hydroxyphenyl)acetyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
3-[1-(3-chloro-4-methylbenzoyl)piperidin-4-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)cyclobutanamine
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[6-(dimethylcarbamoyl)pyrazin-2-yl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1,3-benzothiazole
N-ethyl-1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-3-carboxamide
3-[2-(4-fluorophenyl)azetidine-1-carbonyl]-4-(methoxymethyl)-5-methyl-1,2-oxazole
4-(dimethyl-1,2-oxazol-4-yl)-3-[2-(1H-pyrazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(2,3,6-trimethylphenoxy)acetamide
N-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,1-dimethylpyrrolidin-3-amine
N-[(3S)-2-oxoazepan-3-yl]-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)pyridine-4-carboxamide
2-(3-{[methyl(2,2,6,6-tetramethylpiperidin-4-yl)amino]methyl}-1H-indol-1-yl)acetamide
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-N-ethyl-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N,2-dimethylthieno[2,3-d]pyrimidin-4-amine
methyl 2-({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)pentanoate
2-fluoro-N-({7-[3-(1H-indol-3-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)benzamide
N-[(6-hydroxypyrimidin-4-yl)methyl]-4-(piperidin-3-yl)benzamide
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(4-methyl-1H-imidazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-7-acetamido-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
2-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decane
1-(1-ethyl-1H-pyrazole-4-carbonyl)-3-(3-methylphenyl)piperidine
(2S,4R)-4-amino-1-{3-[(3-hydroxyphenyl)carbamoyl]propanoyl}-N-methylpyrrolidine-2-carboxamide
2-methyl-4-{3-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]phenyl}butan-2-ol
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxylic acid
2-[(4-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenyl)(methyl)amino]ethan-1-ol
1-(2-oxo-2-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethyl)-1,2-dihydropyridin-2-one
2-amino-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-5,6,7,8-tetrahydroquinazoline-4-carboxamide
N,1-dimethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-methyl-N-(1H-pyrazol-3-ylmethyl)-2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
2-benzyl-8-(furan-3-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-2,6-dimethylquinoline
3-{[(cyclopropylcarbamoyl)methyl]sulfamoyl}-N-phenylbenzamide
N-[(4-methoxyphenyl)methyl]-2,4-dimethyl-N-(pyridin-4-ylmethyl)-1,3-oxazole-5-carboxamide
2-(4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
methyl 3-[(3S,4R)-4-(morpholin-4-yl)-1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-3-yl]propanoate
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(ethanesulfonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-({4-[benzyl(methyl)amino]piperidin-1-yl}methyl)pyridine-3-carboxylic acid
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-2-(4-hydroxypiperidin-1-yl)-N-methylacetamide
1-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-4-(2-methylpyridin-4-yl)piperazine
(3aR,6aR)-2-methyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide