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2,3-dimethyl-5-[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]benzene-1-sulfonamide
N-[(5-methylfuran-2-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-({[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
7-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
2-(5-{1-[2-(1H-indazol-3-yl)acetyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetic acid
N-{2-[2-(trifluoromethyl)phenyl]ethyl}-2,3-dihydro-1H-indene-1-carboxamide
N-ethyl-6-methyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
(2S,4R)-1-methyl-N-(propan-2-yl)-4-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamido]pyrrolidine-2-carboxamide
1-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-(1H-imidazol-1-yl)ethan-1-one
(3R,4R)-1-(4-methanesulfonylbenzoyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
3-({[1-(pyridine-4-carbonyl)piperidin-4-yl]amino}methyl)piperidin-3-ol
2-{5-cyclopropyl-4-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-4-(furan-2-yl)pyrimidine
3-(pyrazin-2-yl)-1-{2-[5-(pyrrolidine-1-carbonyl)thiophen-2-yl]pyrrolidin-1-yl}propan-1-one
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]acetamide
(4aR,7aS)-1-(2-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}pyrimidin-4-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
2-(4-{[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}phenyl)ethan-1-amine
2-{2-[(E)-2-phenylethenyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
N-[1-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]pyridine-3-carboxamide
N-cyclohexyl-1-(piperidin-3-ylmethyl)-N-(pyridin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-(3-chlorophenyl)-4-{1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}piperazine
N-({6-[(E)-2-phenylethenyl]pyridin-3-yl}methyl)acetamide
1-{2-[2-(2,2-diphenylethyl)morpholin-4-yl]-2-oxoethyl}pyrrolidin-2-one
3-(1-methyl-1H-imidazole-2-carbonyl)-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
(1S,5R)-6-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][(1-methyl-1H-imidazol-2-yl)methyl]amine
2-(4-methoxy-2-methylphenyl)-5,6-dimethylpyridine-3-carboxamide
N4-methyl-N2-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]pyrimidine-2,4-diamine
1-[(4-fluorophenyl)methyl]-4-(2-methoxypyrimidine-5-carbonyl)-2-(propan-2-yl)-1,4-diazepane
N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-4-methoxybenzamide
{1-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(3-methylbut-2-en-1-yl)piperidin-3-yl}methanol
N-(3,4-difluorophenyl)-5-{1-[(2,4-difluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-1-benzofuran-2-carboxamide
4-(2-{1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]piperidin-2-yl}ethyl)phenol
2-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-1-(morpholin-4-yl)ethan-1-one
2-[1-(2-phenylethyl)-4-(pyridin-2-ylmethyl)piperazin-2-yl]ethan-1-ol
3-[(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)sulfamoyl]-N-(pentan-3-yl)benzamide
methyl 3-{[4-(3-fluorobenzoyl)-7-oxo-1,4-diazepan-1-yl]methyl}benzoate
4-(1-butyl-1H-imidazol-2-yl)-1-(pyrrolidine-1-carbonyl)piperidine
(3S,4S)-1-(2-amino-5-ethyl-6-methylpyrimidin-4-yl)-4-(dimethylamino)pyrrolidin-3-ol
1-(3-methylpyridin-2-yl)-4-[(1-phenyl-1H-pyrazol-5-yl)methyl]piperazine
3-hexyl-8-(trimethyl-1H-pyrazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(1-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
5-[2-(4-chlorophenyl)morpholine-4-carbonyl]-2-methylphenol
4-[1-(1-benzyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]thiomorpholine
5-(morpholin-4-ylmethyl)-N-[(1R)-2,2,2-trifluoro-1-phenylethyl]furan-3-carboxamide
4-phenoxy-1-[(2S)-piperidine-2-carbonyl]piperidine-4-carboxylic acid
(3aR,6aR)-2-(butane-1-sulfonyl)-5-(cyclobutylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[1-(4-chlorophenyl)cyclobutyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-[5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
N-methyl-5-[2-(methylsulfanyl)phenoxymethyl]-N-(1H-pyrazol-3-ylmethyl)-1,2-oxazole-3-carboxamide