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(3R)-1-(6-amino-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)pyrrolidin-3-ol
4-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-fluoropyridine
2-(propan-2-yl)-4-{[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}pyrimidine
(4S)-1-[(3,5-dimethyl-1H-indol-2-yl)methyl]-3,3,4-trimethylpiperidin-4-ol
1-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
1-ethyl-4-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
1-methyl-3-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,2-dihydroquinoxalin-2-one
6-[(diethylamino)methyl]-N-(oxolan-3-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-(4-{[3-(2-methylpropyl)morpholin-4-yl]methyl}phenoxy)ethan-1-ol
2-methoxy-N-{[1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(4-ethylpiperazin-1-yl)acetamide
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(pyrrolidine-1-carbonyl)piperidine
1-[1-(propan-2-yl)piperidine-3-carbonyl]-4-(4H-1,2,4-triazol-3-yl)piperidine
N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-(pyridin-3-yl)piperazine
N-[(4-cyanophenyl)methyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
1-[2-(4-methoxyphenyl)ethyl]-4-{[5-(trifluoromethyl)pyridin-2-yl]amino}pyrrolidin-2-one
(3S,4R)-1-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-N,N-dimethyl-4-propylpyrrolidin-3-amine
N,N-dimethyl-6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrimidin-4-amine
6-chloro-N,N-dimethyl-3-[({[3-(trifluoromethyl)phenyl]methyl}amino)methyl]imidazo[1,2-a]pyridine-2-carboxamide
1-[1-(3-chloro-4-fluorobenzoyl)piperidin-3-yl]-4-(3-chlorophenyl)piperazine
4-(2,6-dimethylquinoline-3-carbonyl)-3-methylpiperazin-2-one
2-(4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-5-fluoropyrimidine
4-{[(3-methoxyphenyl)methyl]amino}-5-methyl-N-(oxolan-3-yl)thieno[2,3-d]pyrimidine-6-carboxamide
5-ethyl-N-(2-methanesulfonamidoethyl)-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
N-[2-(3-methoxyphenyl)-1-[1-(1-methylpiperidine-2-carbonyl)piperidin-4-yl]ethyl]-N-methylpyridine-3-carboxamide
9-[(5-chloro-3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(morpholin-4-yl)ethyl]amine
2-{4-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[(3S,4R)-1-[(4,6-dimethylpyrimidin-2-yl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
2-(4-{[methyl(propan-2-yl)amino]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
1-methyl-4-{[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrazole
{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}[(dimethyl-1,2-oxazol-4-yl)methyl]methylamine
3-[2-(3-fluorophenyl)piperidine-1-carbonyl]-5-methoxy-1H-indazole
[(5-{1-[(dimethyl-1,3-thiazol-5-yl)methyl]-1H-1,2,3-triazol-4-yl}thiophen-3-yl)methyl]dimethylamine
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
6,7-dimethoxy-2-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
(2S,4S)-N-ethyl-1-(4-methylpent-3-en-1-yl)-4-[2-(3-methylphenyl)acetamido]pyrrolidine-2-carboxamide
N-[(3-methoxyphenyl)methyl]-3-{1-[2-(thiophen-2-yl)acetyl]piperidin-3-yl}propanamide
8-(2-aminoacetyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
1-ethenyl-N-methyl-N-[1-(pyridin-3-yl)propyl]-1H-pyrazole-4-carboxamide
1-benzyl-3-(2-methylpropyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
1-{1'-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(dimethylamino)-N-methylbenzamide
1-{3,5-dimethyl-4-[3-(pyridin-3-yl)azetidine-1-carbonyl]-1H-pyrrol-2-yl}ethan-1-one
1-(morpholin-4-yl)-3-(1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidin-4-yl)propan-1-one
3-{2-[(3-hydroxypropyl)[(5-methylthiophen-2-yl)methyl]amino]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one