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3-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
N-{2-[3-(thiophen-2-yl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
2-(4-{[3-(benzyloxy)phenyl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
5-(3-chlorophenyl)-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,2,4-triazin-3-amine
1-(4-methoxyphenyl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)cyclopropane-1-carboxamide
1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-2-(1,3-thiazol-2-yl)piperidine
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-5-oxopyrrolidine-3-carboxamide
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(4-fluoro-3-methoxyphenyl)methyl]amine
N-[2-(1H-indol-1-yl)ethyl]-2-methyl-1,3-benzoxazole-6-carboxamide
3-(4-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)-1,2-benzothiazole
2-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-2-azaspiro[4.5]decan-3-one
1-[2-benzyl-4-(3-methoxyphenyl)-5-oxopiperazin-1-yl]pentane-1,4-dione
6-chloro-3-{pyrazolo[1,5-a]pyrimidin-3-yl}-[1,2,4]triazolo[4,3-a]pyridine
1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-3-(1H-pyrazol-5-yl)piperidine
7-{[(3-methoxypropyl)(1-methylpiperidin-4-yl)amino]methyl}-2-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
6-tert-butyl-1-methyl-N-[4-(methylamino)butyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-ethyl-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)pyrazolo[1,5-a]pyrimidin-7-amine
[(3R,4S)-4-[(4-methylpiperazin-1-yl)methyl]-1-{[2-(trifluoromethoxy)phenyl]methyl}pyrrolidin-3-yl]methanol
[(2S)-1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl]methanol
(4aS,7aR)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-1-methyl-1H-indole
4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-1-[5-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperidine
(4aS,7aR)-1-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(6-methylpyridin-2-yl)-4-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazine
2-(5-{[(1R,5S,6S)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexan-3-yl]methyl}furan-2-yl)benzonitrile
4-{[4-phenyl-5-(2-phenylethyl)-1H-imidazol-1-yl]methyl}pyrimidine
2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-[2-(2,4,6-trimethylphenoxy)ethyl]acetamide
4-(2-ethylphenyl)-7H-pyrrolo[2,3-d]pyrimidine
2-methoxy-1-[1'-(1-methyl-1H-imidazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
8-[3-(5-methylfuran-2-yl)butyl]-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-fluoro-2-{[3-(pyridin-3-yl)azetidin-1-yl]methyl}quinolin-4-ol
4-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}-1,4-oxazepan-5-one
(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methanol
1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-(propan-2-yl)piperazine
2,7-dimethyl-4-(oxane-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1S,5R)-6-(2H-1,3-benzodioxole-5-carbonyl)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane
1-[(4aR,8aR)-7-{[4-ethoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
(3R,4S)-4-{ethyl[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]amino}oxolan-3-ol
7-(cyclohexylmethyl)-2-(1-methylpiperidine-4-carbonyl)-2,7-diazaspiro[4.5]decane
1-{3-oxo-3-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]propyl}-1,2-dihydropyridin-2-one
8-{imidazo[1,2-a]pyrimidine-2-carbonyl}-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
8-[4-chloro-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
5-cyclopropanecarbonyl-1'-[(2,3,4-trifluorophenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(1R)-1-(4-fluorophenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(3aS,6aR)-5-(4,6-dimethoxypyrimidin-2-yl)-3-[(2-methoxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
8-[(3-hydroxyphenyl)methyl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(azepan-1-yl)ethyl]-2-methyl-6-(piperidin-3-yl)pyrimidin-4-amine
(2R,6S)-4-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperidin-4-yl}-2,6-dimethylmorpholine
(1S,5R)-3-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N,8-dimethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide