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1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-(4-methoxy-3,5-dimethylbenzoyl)piperidine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
2-(furan-2-yl)-5-({4-[6-(propan-2-yl)pyridin-2-yl]piperazin-1-yl}methyl)pyrimidine
methyl 5-[4,5-dimethyl-2-(1H-1,2,3,4-tetrazol-1-yl)thiophene-3-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-(3-fluorophenyl)-4-{1H-imidazo[4,5-b]pyridin-2-yl}-3-(5-methylfuran-2-yl)-1H-pyrazole
1-(2,6-dimethylpyridine-4-carbonyl)-4-(4-methoxybutyl)piperazine
3-({1-[(2-aminopyridin-3-yl)methyl]piperidin-4-yl}methyl)benzoic acid
2-(cyclohex-1-en-1-yl)-1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
6-(methoxymethyl)-N,1-dimethyl-N-[(3-methylthiophen-2-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1-(3-methoxypropyl)-4-phenyl-1H-imidazole
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
1-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]-3-(2-methylphenyl)pyrrolidin-3-ol
1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-[(3S)-1-{3-[(2-methylprop-2-en-1-yl)oxy]benzoyl}pyrrolidin-3-yl]acetamide
2,2-dimethyl-N-(1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
6-[2,2-dimethyl-1-(thiophen-2-yl)cyclopropanecarbonyl]-2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-3-(2-methylphenyl)pyrrolidin-3-ol
1-[4-(oxan-2-ylmethoxy)phenyl]-3-[3-(1H-1,2,4-triazol-1-yl)propyl]urea
5-({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}amino)-1-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-[2-(3-fluorophenyl)ethyl]piperidine
1-({2-[2-hydroxy-3-(thiomorpholin-4-yl)propoxy]phenyl}methyl)azetidin-3-ol
1-[(2S)-2-{3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl}pyrrolidin-1-yl]ethan-1-one
1-(6-hydroxy-1,4-diazepan-1-yl)-2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethan-1-one
1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]azepan-3-amine
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-3-(trifluoromethyl)pyridin-2-amine
5-chloro-N-[3-hydroxy-1-(4-methylphenyl)propyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(2S,4S)-4-amino-N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-1-methylpyrrolidine-2-carboxamide
9-[4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}pyrrolidin-3-yl)-3,5-dimethyl-1H-pyrazole
8-{[3-(trifluoromethyl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
3-{1-[(3-acetylphenyl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
1-(cyclohexylmethyl)-N5-[1-(6-methoxynaphthalen-2-yl)ethyl]-N3,N3-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
{[5-(3-chlorophenyl)furan-2-yl]methyl}(methyl){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
3-(5-chloro-2-ethoxyphenyl)-N,N-dimethyl-1H-1,2,4-triazol-5-amine
N-methyl-3-[N-methyl-1-(2,5,7-trimethylquinolin-4-yl)formamido]propanamide
2-hydroxy-3-methyl-1-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]butan-1-one
(2S,3R)-2-{[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]amino}-3-hydroxybutanamide
6-methyl-2-({[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](prop-2-en-1-yl)amino}methyl)pyridin-3-ol
4-ethyl-1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
6-(aminomethyl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}pyrimidin-4-amine
(1S,5R)-3-[(3-hydroxy-4-methoxyphenyl)methyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3R,9aR)-3-(propan-2-yl)-8-(quinolin-8-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N'1-butyl-N'1-[(2-methylphenyl)methyl]cyclopropane-1,1-dicarboxamide
3-(2,3-difluorophenyl)-1-(oxan-3-ylmethyl)urea
(2E)-N-{[4-(but-2-yn-1-yloxy)phenyl]methyl}-3-(2-chlorophenyl)-N-(pyridin-3-ylmethyl)prop-2-enamide
2-amino-4-(1,2-dimethyl-1H-imidazol-5-yl)-6-(4-methoxyphenyl)-5-methylpyridine-3-carbonitrile
3-[5-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)thiophen-3-yl]prop-2-yn-1-ol
N-[(6-methylpyridin-2-yl)methyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
(4aS,8aR)-6-(3-chloro-4-hydroxybenzoyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
3-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-1-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}urea