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5-[(2-ethylpyrimidin-4-yl)methyl]-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(4-fluorophenyl)piperazin-2-one
6-[(1H-1,2,3,4-tetrazol-5-ylmethyl)amino]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
4-[4-(benzyloxy)piperidine-1-carbonyl]-1-methyl-1H-indole
N-(3-{3-[(dimethylamino)methyl]-1,2,4-oxadiazol-5-yl}phenyl)butanamide
1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
5-acetyl-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}thiophene-2-carboxamide
N-{1-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
2-(1H-1,3-benzodiazol-1-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}propanamide
2-amino-7-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(4-{[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]amino}piperidin-1-yl)ethan-1-one
8-[2-(adamantan-1-ylsulfanyl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
3-(3-hydroxy-3-methylbutyl)-N-(2-hydroxyethyl)-N-[(2-methylphenyl)methyl]benzamide
1-(cyclohexylmethyl)-6-oxo-N-[2-(pyridin-3-yl)ethyl]piperidine-3-carboxamide
1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-4-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperazine
[(1-ethyl-1H-imidazol-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(3-methoxypropyl)piperidine-3-carboxamide
3-[2-(azepan-1-yl)ethyl]-1-cyclohexyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
(4aS,7aR)-1-(5-methylpyrazine-2-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(dimethyl-1,2-oxazol-4-yl)-N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
methyl 3-(1H-indazole-3-carbonyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[(4-acetyl-4-phenylpiperidin-1-yl)methyl]benzonitrile
1-[1-(furan-2-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-3-hydroxypropan-1-one
3-(3-hydroxyquinoxalin-2-yl)-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}propan-1-one
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-3-(2-methoxyphenyl)propanamide
4-[4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carbonyl]-N,N-dimethylpiperazine-1-carboxamide
(4aS,8aR)-6-(2-aminoacetyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
ethyl 5-(cyclohex-3-ene-1-carbonyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[4-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
methyl 4-{[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}butanoate
2-(4-{[3-(methylsulfanyl)phenyl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
2-(furan-2-yl)-1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}azepane
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-(5-propylpyrimidin-4-yl)pyrrolidin-3-yl]methanol
(2S,4R)-4-({[3-(benzyloxy)phenyl]methyl}amino)-1-[(2-chlorophenyl)methyl]-N-ethylpyrrolidine-2-carboxamide
8-[(1-ethyl-1H-indol-4-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
6-(4-fluorophenyl)-N-(3-hydroxypropyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
methyl({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl){[3-(trifluoromethyl)phenyl]methyl}amine
N-cyclooctyl-6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
4-ethyl-3-{1-[(2E)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enoyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-amino-6-[4-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperazin-1-yl]pyrimidin-4-ol
1-cyclohexanecarbonyl-N-[3-(1H-1,2,4-triazol-1-yl)propyl]pyrrolidine-2-carboxamide
(3S)-1-(1-methyl-5-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1H-1,3-benzodiazol-2-yl)pyrrolidin-3-ol
(3aS,6aS)-2-[(4-methanesulfonylphenyl)methyl]-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1S,5R)-3-(oxan-4-yl)-6-(5-phenyl-1,2-oxazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
7-(2-cyclohexylethyl)-2-(1-methyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-(3-ethoxy-2-hydroxypropyl)-6,8-dimethyl-3,4-dihydroquinazolin-4-one
4-(3-methoxybenzenesulfonyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{[5-(4-methylphenyl)-1,2-oxazol-3-yl]methyl}acetamide
2-[(3,5-difluorophenyl)methyl]-8-(propane-1-sulfonyl)-2,8-diazaspiro[4.5]decan-3-one