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1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-3-(propoxymethyl)pyrrolidine
2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-N-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
2-{[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzonitrile
4-chloro-1,3-dimethyl-N-[3-(4-methylpiperazin-1-yl)propyl]-1H-pyrazole-5-carboxamide
1-[4-({2-[4-(1H-imidazol-1-yl)butoxy]phenyl}methyl)piperazin-1-yl]-2,2-dimethylpropan-1-one
4,6-dimethyl-1-{2-[(4-phenylbutan-2-yl)amino]ethyl}-1,2-dihydropyrimidin-2-one
1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-{[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}-1,3-benzothiazole
6-(4-{[3-(1H-indazol-1-yl)propyl]amino}piperidin-1-yl)pyridine-3-carbonitrile
7-[2-(dimethyl-1,3-thiazol-4-yl)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-{3-[2-(4-fluorophenyl)piperidin-1-yl]-3-oxopropyl}azepan-2-one
5,6-dimethyl-2-[4-({methyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
4-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}pyridine-2-carboxylic acid
N-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
6-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)pyridine-2-carboxylic acid
1-(cyclohexylmethyl)-5-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}piperidin-2-one
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetamide
3-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-4-phenylpyrrolidin-2-one
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
methyl 4-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}(methyl)carbamoyl)benzoate
N-(2-{7-[(4-ethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
3-(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-(2-hydroxyethyl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]urea
N-[(1-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidin-3-yl)methyl]furan-2-carboxamide
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-[4-(3-phenylbutyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
8-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
2-{6-[(2-hydroxyethyl)(methyl)amino]pyridazin-3-yl}benzoic acid
1-[4-(2-amino-5-ethylpyrimidin-4-yl)piperazin-1-yl]ethan-1-one
8-[(3-methoxyphenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(4-benzyl-1H-1,2,3-triazol-1-yl)-1-(furan-3-carbonyl)piperidine
[1-(1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)piperidin-4-yl]methanol
3-(3,4-dimethoxyphenyl)-1-(5-{[(dimethylsulfamoyl)amino]methyl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl)propan-1-one
5-[(2E)-but-2-en-2-yl]-1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4-phenyl-1H-imidazole
4-{1-[5-(4-chloro-3,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}pyridine
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]piperidine-3-carboxamide
1-(6-aminopyridine-3-carbonyl)-N,N-dimethylazepan-4-amine
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
1-[(1-ethylpiperidin-3-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(benzyloxy)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}acetamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2-(2,5-dimethylphenyl)ethyl]-1H-pyrazole-3-carboxamide
N,N-dimethyl-2-(1-{[(1-methyl-1H-indazol-3-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)pyridine-3-carboxamide
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-5-(3-fluorophenyl)-1,2,4-triazin-3-amine
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(3-methoxyphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[(3R,4S)-3-[3-(2-methoxyphenyl)propanamido]-4-(propan-2-yl)pyrrolidin-1-yl]acetic acid
(1S,5R)-3-(3-phenylpropyl)-6-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}({imidazo[1,2-a]pyridin-3-ylmethyl})methylamine
2-(2H-1,3-benzodioxol-5-yl)-1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-fluoro-1H-1,3-benzodiazole
[(3R,4R)-1-[(2,6-difluorophenyl)methyl]-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
N-(1-methyl-1H-1,3-benzodiazol-6-yl)azocane-1-carboxamide
1-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine