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1-(3-fluoro-2-methoxybenzoyl)-3-(hydroxymethyl)piperidin-3-ol
N-[(2-chlorophenyl)methyl]-N-(2-hydroxyethyl)-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
1-[5-methoxy-2-({[3-(methylsulfanyl)propyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
5-(morpholin-4-ylmethyl)-N-(2-oxoazepan-3-yl)furan-3-carboxamide
5-[(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)carbamoyl]-2,1,3-benzoxadiazol-1-ium-1-olate
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N-(butan-2-yl)-N-cyclopentyl-3-(pyridin-3-yl)propanamide
7-cyclohexyl-2-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-(1-{[2-(carbamoylmethoxy)-5-chlorophenyl]methyl}piperidin-3-yl)-N,N-dimethylpropanamide
2-methyl-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-4-phenylpyridine-3-carboxamide
N-cyclohexyl-2-cyclopropyl-N-[2-(ethylsulfanyl)ethyl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
1-methyl-4-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperazin-2-one
2-methyl-8-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
6-{3-[methyl(phenyl)amino]propyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
3-{[3-(trifluoromethoxy)phenyl]methyl}-1,3-oxazolidin-2-one
1-methyl-4-{5-[2-(5-methylfuran-2-yl)phenyl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}piperidine
5-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-3-(2-methylpropyl)-1H-pyrazole
4-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
N-cyclopropyl-3-[1-(2,2-diphenylethyl)piperidin-3-yl]propanamide
N-cyclohexyl-3-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)propanamide
2-{4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenoxy}acetamide
(1S,5R)-3-[(2-fluoro-4-methoxyphenyl)methyl]-3,9-diazabicyclo[3.3.2]decan-10-one
4-[(2,3-difluoro-6-methoxyphenyl)methyl]-2,2-dimethylmorpholine
2-[6-methyl-2-(methylamino)pyrimidin-4-yl]-N,N-bis(propan-2-yl)benzamide
3-(2-methoxyethyl)-1-(2-phenylethyl)piperidine-3-carboxylic acid
N-[(1S,2R)-2-(cyclohexylamino)cyclobutyl]-2-phenoxybenzamide
2-[1-(thiophen-2-ylmethyl)-4-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
2-[3-(2-fluoro-4-methylphenyl)-1H-indazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
7-methyl-3-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-3,7,11-triazaspiro[5.6]dodecan-12-one
1-[(5-ethylfuran-2-yl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
N-[2-(4-fluorobenzenesulfonyl)ethyl]-2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carboxamide
N-[(1R,3R)-3-aminocyclopentyl]-3-(3-methylphenyl)-1H-pyrazole-4-carboxamide
2-butanoyl-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(2-methoxyethyl)(propan-2-yl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
3-ethoxy-N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-4-(prop-2-en-1-yloxy)benzamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamide
1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-3-(1-methyl-1H-imidazol-2-yl)piperidine
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-{[(2-hydroxyethyl)(methyl)amino]methyl}piperidin-2-one
methyl (2S,4R)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(3-methylphenyl)methyl]pyrrolidine-2-carboxylate
2-(1-ethylpiperidin-4-yl)-N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methylacetamide
4-{4-[(4-benzyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-6-methylpyrimidin-2-amine
3-(1H-indol-3-yl)-1-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}propan-1-one
N-{[1-(phenoxymethyl)cyclopropyl]methyl}thian-4-amine
4-({[(2-methoxyphenyl)methyl](propyl)amino}methyl)-N-methylbenzene-1-sulfonamide
methyl({[6-(3-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl})(1,2-oxazol-5-ylmethyl)amine
1-(4-{[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
2-(4-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenyl)-5,6-dimethyl-3,4-dihydropyrimidin-4-one
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-2-{octahydropyrrolo[1,2-a]piperazin-2-yl}pyridine