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N-{[5,8-dimethoxy-2-(4-methylphenyl)quinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
2-(4-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxy)acetic acid
4-({5-[1-(6-methoxypyrimidin-4-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-(4-{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}piperazin-1-yl)ethan-1-ol
4-fluoro-3-{6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}benzene-1-sulfonamide
5-(1-{4-[(methylcarbamoyl)methyl]phenyl}-1H-imidazol-2-yl)thiophene-2-carboxylic acid
7-methoxy-3-{[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
4-methyl-N-[(3R,5S)-1-(pent-2-yn-1-yl)-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]-1H-imidazole-2-carboxamide
3-{[3-phenyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-4-(propan-2-yl)piperazin-2-one
3-(azocan-1-yl)-N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methylpropanamide
2-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]-N,N-bis(prop-2-en-1-yl)acetamide
2-(3-methoxypropyl)-8-(5-propylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
(4aR,8aR)-2-cyclopentanecarbonyl-7-[(5-fluoro-2-methoxyphenyl)methyl]-decahydro-2,7-naphthyridin-4a-ol
N-[1-(cyclohex-1-en-1-yl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
5,7-dimethyl-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]pyrido[2,3-d]pyrimidin-4-amine
5-ethyl-N-[1-methyl-6-(propan-2-yloxy)-1H-indazol-3-yl]thiophene-3-carboxamide
4-(cyclobutylsulfamoyl)-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]benzamide
2-methyl-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4,4-difluoro-1-[4-(1H-imidazol-1-yl)benzoyl]piperidine
N,3,5,7-tetramethyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1H-indole-2-carboxamide
{1-[1-(1-benzylpiperidin-4-yl)piperidine-3-carbonyl]piperidin-4-yl}methanol
2-[(1S,5R)-6-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
9-(2-{[(3,5-dimethylphenyl)methyl]sulfanyl}acetyl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
N,N,4-trimethyl-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyrimidin-2-amine
1-[2-(4-fluorophenyl)ethyl]-4-{[(4-methoxyphenyl)methyl]amino}pyrrolidin-2-one
2-[4-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]pyrazine
(1S,5R)-3-[1-(2-chlorophenyl)piperidin-4-yl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
9-(1-tert-butyl-1H-pyrrole-3-carbonyl)-2-(cyclopropylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[4-(3-methylphenyl)piperazin-1-yl]-1-(5,6,7,8-tetrahydro-1,6-naphthyridin-6-yl)propan-1-one
2-({[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]amino}methyl)-5,8-dimethylquinolin-4-ol
2-(azepan-1-yl)-N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)acetamide
2-amino-6-tert-butyl-4-(2,6-dimethoxyphenyl)pyridine-3-carbonitrile
N-benzyl-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
N-benzyl-4-(2-methoxyphenoxy)piperidine-1-sulfonamide
N-[3-(2-fluorophenyl)propyl]-2-methyl-4-phenylpyrimidine-5-carboxamide
4-({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)piperazin-2-one
6-(3-chlorophenyl)-N-(1-methoxypropan-2-yl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-(5-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-2-chloro-6-fluorobenzamide
1-(4-chlorophenyl)-N-({1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-(1-phenylbutyl)benzamide
1-{3-oxo-3-[4-(pyridin-3-yl)piperazin-1-yl]propyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
methyl 2-[ethyl(2-methylprop-2-en-1-yl)sulfamoyl]-6-(3-fluorobenzoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-chloro-6-[2-(piperidin-1-ylmethyl)phenoxy]pyridazine
N,1-dimethyl-3-propyl-N-(quinoxalin-2-ylmethyl)-1H-pyrazole-5-carboxamide
2-{[5-(2-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}-N,2-dimethylpropanamide
(1R,5R)-6-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3,4,7-trimethyl-2-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]-1H-indole
3-hydroxy-1-(2-methoxyethyl)-3-{[4-(pyridin-4-ylmethyl)piperazin-1-yl]methyl}piperidin-2-one
methyl (2R,4S)-4-hydroxy-1-[4-(2-methylphenyl)benzoyl]piperidine-2-carboxylate
2-{5-[5-(hydroxymethyl)furan-2-yl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol