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3-hydroxy-3-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}-1-(3-phenylpropyl)piperidin-2-one
2-(4-{[2-(3-methylphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}morpholin-2-yl)ethan-1-ol
2-cyclopropyl-9-(3-hydroxypropanoyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
3-{1-[2-(2-methylphenyl)benzoyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
8-[(4-methyl-3,4-dihydro-2H-1,4-benzoxazin-7-yl)sulfonyl]-2,8-diazaspiro[4.5]decan-3-one
5-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-({[(1-cyclopentylpiperidin-4-yl)methyl](pyridin-3-ylmethyl)amino}methyl)phenol
3-methyl-8-(5-propylfuran-2-yl)-2H,3H,5H,6H,7H,8H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione
3-(azocan-1-yl)-N-ethyl-N-(pyridin-4-ylmethyl)propanamide
2-(1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)-1H-1,3-benzodiazole
N-benzyl-2-[(1S,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
2-chloro-5-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]carbamoyl}amino)-N-(propan-2-yl)benzamide
[(3R,4S)-4-(morpholin-4-ylmethyl)-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl]methanol
2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]acetamide
N,4-dimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]-3-(2-oxoimidazolidin-1-yl)benzamide
1-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-phenyl-1,3-thiazol-4-yl)ethan-1-one
methyl 4-{[1-ethyl-2,4-dioxo-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}benzoate
1-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-phenylethan-1-one
N-(2-cyclopropylphenyl)-3-hydroxy-3-phenylpyrrolidine-1-carboxamide
4-(hydroxymethyl)-3-{[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl}-1,3-oxazolidin-2-one
3-(oxan-4-yl)-1-phenyl-5-[(2R)-pyrrolidin-2-yl]-1H-1,2,4-triazole
2-{4-[4-(2,2,2-trifluoroethyl)piperazine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
5-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-N-methylpyrimidin-2-amine
2-methyl-8-(2-propoxybenzoyl)-2,8-diazaspiro[4.5]decane
2-({4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
N-[2-(3-chlorophenoxy)ethyl]-2-(4,4-dimethyl-2-oxopyrrolidin-1-yl)-N-ethylacetamide
{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl){[3-(methylsulfanyl)phenyl]methyl}amine
5-[3-(3-methoxypropyl)piperidine-1-carbonyl]-4-methylpyrimidine
3-{2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}-5-methylpyridine
1-(2-chloro-5-sulfamoylphenyl)-3-[2-(ethylsulfanyl)ethyl]urea
1-(4-{[2-(azepan-1-yl)-2-phenylethyl]amino}piperidin-1-yl)-2-methylpropan-1-one
(3S,4R)-4-(2-methylphenyl)-1-[3-(pyridin-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidine-3-carboxylic acid
N-{[1-(2-methylphenyl)pyrrolidin-3-yl]methyl}-1-(propan-2-yl)piperidine-4-carboxamide
2-{[4-(3-ethenylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-(propan-2-yl)-1H-imidazole
5-{[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-(5-hydroxy-1,2-dimethyl-1H-indole-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
methyl 3-[(benzylsulfamoyl)amino]-4-methylbenzoate
3-(5-cyclobutyl-1,3,4-thiadiazol-2-yl)-1-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]urea
2-chloro-6-methoxy-4-{[3-(morpholin-4-yl)piperidin-1-yl]methyl}phenol
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(3-hydroxypropyl)-N-methylpropanamide
4-(2-fluoro-5-methylphenoxy)-1-(oxolane-3-carbonyl)piperidine-4-carboxylic acid
2-[1-(1-cyclopropylethyl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-6-ethoxyphenol
1-cyclopentyl-4-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperazin-2-one
N-cyclopropyl-3-[5-(3-methanesulfonylpropanoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
1-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-5-phenyl-1H-pyrrole-2-carboxamide
N-[(3-chlorophenyl)methyl]-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
5-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-(pyridin-3-yl)furan-2-carboxamide
3-{6-amino-5-cyano-4-[3-(1H-pyrazol-1-yl)phenyl]pyridin-2-yl}-1H-pyrazole-5-carboxylic acid