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4-[1-(3-fluorophenyl)-5-(2-methanesulfonylethyl)-1H-1,2,4-triazol-3-yl]pyridine
3-{5-[1-(4-chloro-1H-pyrazol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
N-[1-(6-methylpyridin-3-yl)ethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(2R,3R)-3-amino-1'-(4-propylpyrimidine-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
5-(cyclopentylamino)-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-N-(propan-2-yl)pyridine-4-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(4-methoxyphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(2H-1,3-benzodioxol-5-yl)-1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperidin-3-amine
5-methyl-1'-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl({[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
4-{2-methyl-6-[1-(4-methyl-1H-imidazole-5-carbonyl)piperidin-3-yl]pyrimidin-4-yl}morpholine
N-methyl-2-[methyl({[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl})amino]acetamide
1-(4-{7-chloro-3-[({[3-(trifluoromethyl)phenyl]methyl}amino)methyl]quinolin-2-yl}piperazin-1-yl)ethan-1-one
1-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
methyl 4-[({1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]piperidin-4-yl}amino)methyl]benzoate
1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
6-{[1-(furan-2-yl)ethyl]amino}-N-methyl-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
methyl 4-({2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]acetamido}methyl)benzoate
8-(2-methoxypyridine-3-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(2-methylpyridin-4-yl)piperazine
4-[5-(methoxymethyl)furan-2-carbonyl]-1-[(4-methoxyphenyl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
4-phenyl-N-{[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-3-yl]methyl}benzamide
1-(azepan-1-yl)-3-{3-[(tert-butylamino)methyl]phenoxy}propan-2-ol
3-(2-fluorophenyl)-5-(thiophen-2-ylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
(4aS,8aR)-6-(5-chloro-3-fluoropyridin-2-yl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
5-{[(4-methanesulfonylmorpholin-2-yl)methyl]carbamoyl}thiophene-2-carboxylic acid
methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
N-(2,3-dihydro-1H-inden-1-yl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
6-(3-chlorophenyl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[3-hydroxy-1-(4-methylphenyl)propyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-{2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
N-(2-hydroxyethyl)-1-[1-(6-methylpyridine-2-carbonyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
1-tert-butyl-4-{1-butyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-3,5-dimethyl-1H-pyrazole
3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-[2-methyl-5-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
2-methyl-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-(4-methyl-1,4-diazepane-1-carbonyl)-6-(thiophen-2-ylmethyl)-6-azaspiro[2.5]octane
5-methyl-3-{2-oxo-2-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethyl}-2,3-dihydro-1H-indol-2-one
2-(3-methoxyphenyl)-N-methyl-N-(propan-2-yl)-1,3-benzoxazole-6-carboxamide
2-(4-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-oxo-2H-chromene-3-carboxamide
N-[1-(3-hydroxyadamantan-1-yl)ethyl]-2-methoxypyrimidine-5-carboxamide
1-ethyl-3-(piperidine-1-carbonyl)-N,N-bis(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-[4-(piperidine-1-carbonyl)phenyl]urea
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenoxy]-N-cyclopentylacetamide
3-(4-methyl-1,3-thiazol-5-yl)-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}propanamide
1-({3-[2-(methylsulfanyl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}methyl)piperidin-2-one