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5-cyclobutanecarbonyl-1'-(dimethyl-1,2-oxazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(6-methoxy-2H-chromen-3-yl)methyl]-3-(1H-pyrazol-5-yl)piperidine
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(4-phenylphenyl)methyl]amino}pyrrolidine-2-carboxamide
N,N-dimethyl-2-({[2-(methylsulfanyl)pyrimidin-4-yl]amino}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
5-{4-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
4-{1-[1-butyl-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}morpholine
N,6-dimethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-2-(morpholin-4-yl)pyrimidin-4-amine
2-methyl-4-{3-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]phenyl}butan-2-ol
3-(5-{[4-(5-chloropyrimidin-2-yl)piperazin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
4-[(1H-imidazol-2-ylmethyl)sulfamoyl]-N-(pyridin-2-ylmethyl)benzamide
6-chloro-8-methyl-4-[2-(trifluoromethyl)morpholin-4-yl]quinoline
(2S)-2-{[(2,5-dimethylthiophen-3-yl)methyl]amino}-3-phenylpropanamide
2-(1,5-dimethyl-1H-indole-2-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
(2S,4R)-1-[(3,4-difluorophenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]-N-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
5-(2-ethylbenzoyl)-1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
N3-[2-(3-chlorophenyl)ethyl]-N5-[(3-fluorophenyl)methyl]-1-(2-methoxyethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)urea
(3aS,6aR)-3-cyclopentyl-5-{7-methylthieno[3,2-d]pyrimidin-4-yl}-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
dimethyl[3-(4-{[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl}phenoxy)propyl]amine
6-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepin-3-one
[(3R,4R)-1-(2,3-dihydro-1,4-benzodioxine-5-sulfonyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
ethyl 1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(2-phenoxyethyl)piperidine-3-carboxylate
(1S,6R)-9-[2-(4-ethylphenoxy)acetyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-[3-({4-[(3-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)phenoxy]ethan-1-ol
3-(3-chlorophenyl)-3-(3-hydroxyphenyl)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]propanamide
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2,6-dimethylquinoline-3-carboxamide
4-[(dipropylamino)methyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]benzamide
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3-(pyrrolidin-3-yl)benzamide
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(furan-2-yl)propanamide
N-[(3R,4S)-4-cyclopropyl-1-(1-phenylcyclopropanecarbonyl)pyrrolidin-3-yl]methanesulfonamide
N-cyclopropyl-3-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}propanamide
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}butane-1-sulfonamide
4-chloro-1-methyl-3-({4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)-1H-indazole
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
N-(adamantan-1-yl)-6-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
ethyl 1-ethyl-5-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(3R,4R)-3-cyclopropyl-1-{[1-(methoxymethyl)-1H-imidazol-2-yl]methyl}-4-methylpyrrolidin-3-ol
methyl 1-benzyl-5-{[(2,3-dimethoxyphenyl)methyl]amino}-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-chloro-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-1,3-dimethyl-1H-indole-2-carboxamide
(1S,9R)-11-[(6-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
2-amino-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)-4-[2-(prop-2-en-1-yloxy)phenyl]pyridine-3-carbonitrile
3-[(4-fluorophenyl)formamido]-N-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}propanamide
N-[(3S,4R)-4-propyl-1-(9H-purin-6-yl)pyrrolidin-3-yl]acetamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
(2S,4R)-4-amino-N-ethyl-1-[2-(methylsulfanyl)pyridine-3-carbonyl]pyrrolidine-2-carboxamide
6-[(3-methoxypiperidin-1-yl)methyl]-1-methyl-1H-indole
2-chloro-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]-5-(1H-pyrazol-1-yl)benzamide