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(1R,3S)-3-[cyclopropyl(1H-indol-5-ylmethyl)carbamoyl]cyclopentane-1-carboxylic acid
N-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-3-(2-fluorophenyl)pyrrolidine-1-carboxamide
1-(4-methylquinazolin-2-yl)-N-(oxan-4-ylmethyl)piperidine-4-carboxamide
5-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1H-1,2,3-triazol-4-yl}pyrimidine
2-cyclohexyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-benzoxazole-6-carboxamide
3-({1-[3-(methylsulfanyl)propyl]piperidin-4-yl}oxy)-N-(2-phenylethyl)benzamide
2-(2-aminoethyl)-N-[2-(morpholin-4-yl)ethyl]quinazolin-4-amine
2-methyl-3-({4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)quinoxaline
3-{1-[(2R)-2-amino-3-(ethylsulfanyl)propanoyl]piperidin-4-yl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(3aS,6aR)-3-[2-(pyridin-2-yl)ethyl]-5-(pyridin-3-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N,N-dimethyl-5-[2-(methylamino)pyridine-3-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-{[(5-ethylpyridin-2-yl)methyl]sulfamoyl}-N-(propan-2-yl)benzamide
(4aS,7aR)-1-[3-(4-hydroxyphenyl)propanoyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(propan-2-yloxy)ethan-1-one
2-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-4H-chromen-4-one
5-fluoro-N-(2-methoxyethyl)-N-[(3-methoxyphenyl)methyl]-1,3-dimethyl-1H-indole-2-carboxamide
1-(4-{[(2S)-2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
1-(3-chlorophenyl)-4-[(3-{2-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl]piperazine
8-methoxy-3-[2-(4-methylpiperazin-1-yl)ethyl]-3,4-dihydroquinazolin-4-one
1-cyclohexyl-N3,N5-dimethyl-4-oxo-N3-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-(2,4-dimethylphenoxy)ethyl]-N-methyl-2-(morpholin-4-yl)pyridine-3-carboxamide
3-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-2-methyl-4,5,6,7-tetrahydro-2H-indazole
4-[2-chloro-5-(pyrrolidine-1-carbonyl)phenyl]-4H-1,2,4-triazole
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-(trifluoromethyl)pyrimidin-2-amine
N-[(2,5-difluorophenyl)methyl]-N'-(2-methylphenyl)propanediamide
N-cyclobutyl-4-(1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
5-(8-methoxy-2-methylquinolin-5-yl)pyridin-2-amine
1-(1-methyl-3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-1,2,4-triazol-5-yl)piperidine
(1R,3S)-3-({2-[ethyl(3-methylphenyl)amino]ethyl}carbamoyl)cyclopentane-1-carboxylic acid
N-{4-[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]-4-oxobutyl}acetamide
2-[(3R,4R)-3-hydroxy-4-(pyrazine-2-amido)piperidin-1-yl]-6-methylpyridine-3-carboxylic acid
5-fluoro-N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)quinazolin-4-amine
N-[2-(1H-imidazol-4-yl)ethyl]-N'-(2,4,6-trimethylphenyl)butanediamide
3-(2-methylpropyl)-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-oxazole-5-carboxamide
1,5-dimethyl-4-{[3-(naphthalene-1-carbonyl)piperidin-1-yl]methyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
5-(azepane-1-carbonyl)-1-(butan-2-yl)-4-oxo-N-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2,6-dimethyl-4-[4-(oxolan-2-ylmethyl)piperazine-1-carbonyl]quinoline
1-[3-(2-ethyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-3-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}urea
1-(morpholin-4-yl)-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
4-{1-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]azetidin-3-yl}morpholine
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
2,3-dimethyl-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]quinoxaline-6-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-propyl-N-(pyridin-3-ylmethyl)acetamide
N-[(6-oxo-1,6-dihydropyrimidin-4-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
methyl 5-[(3-methylbutyl)amino]-3-(oxolane-3-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
6-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]-1,2-dihydropyridin-2-one
1-{3-[(3S,4S)-3,4-dihydroxypiperidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-hydroxy-1-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]ethan-1-one
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(oxan-4-ylmethyl)amine